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Increased number of cardiac adrenergic receptors following local heart irradiation

Journal Article · · Radiation Research; (USA)
DOI:https://doi.org/10.2307/3577375· OSTI ID:5600979
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  1. Institut fuer Strahlenbiologie, Neuherberg (Germany, F.R.)
The effect of local X irradiation on cardiac alpha and beta receptors was studied in Wistar rats. Animals were given local heart irradiation with single doses of 15 or 20 Gy and were examined after a range of latency times of 7 to 400 days. Using the radioactive ligands ({sup 3}H)CGP-12177 and ({sup 3}H)prazosin, the maximal binding capacity was determined from saturation experiments. At 7 days after 20 Gy the maximal binding capacity of both alpha and beta receptors was reduced to below the level of untreated control animals. Subsequently it rose continually to a maximum of 160% of the control level for beta receptors and 130% for alpha receptors at 400 days postirradiation. The antagonist affinity as judged from the dissociation constant for ({sup 3}H)CGP 12177 and ({sup 3}H)prazosin did not change significantly. A similar effect was observed after 15 Gy. An increase in adrenergic receptors may represent an important pathogenetic link between early morphological and late functional changes in the pathogenesis of radiation-induced heart disease.
OSTI ID:
5600979
Journal Information:
Radiation Research; (USA), Journal Name: Radiation Research; (USA) Vol. 119:1; ISSN RAREA; ISSN 0033-7587
Country of Publication:
United States
Language:
English