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Synthesis of 4-substituted-trans-1,2-diaminocyclohexyl polyaminocarboxylate metal chelating agents for the preparation of stable radiometal antibody immunoconjugates for therapy and SPECT and PET imaging

Patent ·
OSTI ID:489096

Cyclohexyl chelating agents useful in forming antibody-metal conjugates which are used for diagnostic and therapeutic purposes are synthesized. New compounds and processes of forming these compounds are disclosed including 4-haloacetamido-trans-1,2-diaminocyclohexyl polyaminocarboxylate and 4-isothiocyanato-trans-1,2-diamino cyclohexane-N,N,N{prime},N{prime}-tetra acetic acid.

Research Organization:
Associated Universities Inc
Sponsoring Organization:
USDOE, Washington, DC (United States)
DOE Contract Number:
AC02-76CH00016
Assignee:
PTO; 550604; SN: 97001799038; SCA: 550601; PA: EDB-97:087810
Patent Number(s):
US 5,635,157/A/
Application Number:
PAN: 8-132,201
OSTI ID:
489096
Country of Publication:
United States
Language:
English