Optimization of a binding fragment targeting the “enlarged methionine pocket” leads to potent Trypanosoma brucei methionyl-tRNA synthetase inhibitors
- Authors:
- Publication Date:
- Sponsoring Org.:
- USDOE Office of Science (SC), Basic Energy Sciences (BES)
- OSTI Identifier:
- 1416585
- Grant/Contract Number:
- AC02-76SF00515
- Resource Type:
- Publisher's Accepted Manuscript
- Journal Name:
- Bioorganic and Medicinal Chemistry Letters
- Additional Journal Information:
- Journal Name: Bioorganic and Medicinal Chemistry Letters Journal Volume: 27 Journal Issue: 12; Journal ID: ISSN 0960-894X
- Publisher:
- Elsevier
- Country of Publication:
- United Kingdom
- Language:
- English
Citation Formats
Huang, Wenlin, Zhang, Zhongsheng, Ranade, Ranae M., Gillespie, J. Robert, Barros-Álvarez, Ximena, Creason, Sharon A., Shibata, Sayaka, Verlinde, Christophe L. M. J., Hol, Wim G. J., Buckner, Frederick S., and Fan, Erkang. Optimization of a binding fragment targeting the “enlarged methionine pocket” leads to potent Trypanosoma brucei methionyl-tRNA synthetase inhibitors. United Kingdom: N. p., 2017.
Web. doi:10.1016/j.bmcl.2017.04.048.
Huang, Wenlin, Zhang, Zhongsheng, Ranade, Ranae M., Gillespie, J. Robert, Barros-Álvarez, Ximena, Creason, Sharon A., Shibata, Sayaka, Verlinde, Christophe L. M. J., Hol, Wim G. J., Buckner, Frederick S., & Fan, Erkang. Optimization of a binding fragment targeting the “enlarged methionine pocket” leads to potent Trypanosoma brucei methionyl-tRNA synthetase inhibitors. United Kingdom. https://doi.org/10.1016/j.bmcl.2017.04.048
Huang, Wenlin, Zhang, Zhongsheng, Ranade, Ranae M., Gillespie, J. Robert, Barros-Álvarez, Ximena, Creason, Sharon A., Shibata, Sayaka, Verlinde, Christophe L. M. J., Hol, Wim G. J., Buckner, Frederick S., and Fan, Erkang. Thu .
"Optimization of a binding fragment targeting the “enlarged methionine pocket” leads to potent Trypanosoma brucei methionyl-tRNA synthetase inhibitors". United Kingdom. https://doi.org/10.1016/j.bmcl.2017.04.048.
@article{osti_1416585,
title = {Optimization of a binding fragment targeting the “enlarged methionine pocket” leads to potent Trypanosoma brucei methionyl-tRNA synthetase inhibitors},
author = {Huang, Wenlin and Zhang, Zhongsheng and Ranade, Ranae M. and Gillespie, J. Robert and Barros-Álvarez, Ximena and Creason, Sharon A. and Shibata, Sayaka and Verlinde, Christophe L. M. J. and Hol, Wim G. J. and Buckner, Frederick S. and Fan, Erkang},
abstractNote = {},
doi = {10.1016/j.bmcl.2017.04.048},
journal = {Bioorganic and Medicinal Chemistry Letters},
number = 12,
volume = 27,
place = {United Kingdom},
year = {Thu Jun 01 00:00:00 EDT 2017},
month = {Thu Jun 01 00:00:00 EDT 2017}
}
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https://doi.org/10.1016/j.bmcl.2017.04.048
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Cited by: 13 works
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