Structure-Guided Development of Deoxycytidine Kinase Inhibitors with Nanomolar Affinity and Improved Metabolic Stability
- Authors:
-
- Department of Biochemistry and Molecular Genetics, and ‡Center for Pharmaceutical Biotechnology, University of Illinois at Chicago, Chicago, Illinois 60607, United States
- Publication Date:
- Sponsoring Org.:
- USDOE
- OSTI Identifier:
- 1163572
- Grant/Contract Number:
- AC02- 06CH11357
- Resource Type:
- Published Article
- Journal Name:
- Journal of Medicinal Chemistry
- Additional Journal Information:
- Journal Name: Journal of Medicinal Chemistry Journal Volume: 57 Journal Issue: 22; Journal ID: ISSN 0022-2623
- Publisher:
- American Chemical Society
- Country of Publication:
- United States
- Language:
- English
Citation Formats
Nomme, Julian, Li, Zheng, Gipson, Raymond M., Wang, Jue, Armijo, Amanda L., Le, Thuc, Poddar, Soumya, Smith, Tony, Santarsiero, Bernard D., Nguyen, Hien-Anh, Czernin, Johannes, Alexandrova, Anastassia N., Jung, Michael E., Radu, Caius G., and Lavie, Arnon. Structure-Guided Development of Deoxycytidine Kinase Inhibitors with Nanomolar Affinity and Improved Metabolic Stability. United States: N. p., 2014.
Web. doi:10.1021/jm501124j.
Nomme, Julian, Li, Zheng, Gipson, Raymond M., Wang, Jue, Armijo, Amanda L., Le, Thuc, Poddar, Soumya, Smith, Tony, Santarsiero, Bernard D., Nguyen, Hien-Anh, Czernin, Johannes, Alexandrova, Anastassia N., Jung, Michael E., Radu, Caius G., & Lavie, Arnon. Structure-Guided Development of Deoxycytidine Kinase Inhibitors with Nanomolar Affinity and Improved Metabolic Stability. United States. https://doi.org/10.1021/jm501124j
Nomme, Julian, Li, Zheng, Gipson, Raymond M., Wang, Jue, Armijo, Amanda L., Le, Thuc, Poddar, Soumya, Smith, Tony, Santarsiero, Bernard D., Nguyen, Hien-Anh, Czernin, Johannes, Alexandrova, Anastassia N., Jung, Michael E., Radu, Caius G., and Lavie, Arnon. Fri .
"Structure-Guided Development of Deoxycytidine Kinase Inhibitors with Nanomolar Affinity and Improved Metabolic Stability". United States. https://doi.org/10.1021/jm501124j.
@article{osti_1163572,
title = {Structure-Guided Development of Deoxycytidine Kinase Inhibitors with Nanomolar Affinity and Improved Metabolic Stability},
author = {Nomme, Julian and Li, Zheng and Gipson, Raymond M. and Wang, Jue and Armijo, Amanda L. and Le, Thuc and Poddar, Soumya and Smith, Tony and Santarsiero, Bernard D. and Nguyen, Hien-Anh and Czernin, Johannes and Alexandrova, Anastassia N. and Jung, Michael E. and Radu, Caius G. and Lavie, Arnon},
abstractNote = {},
doi = {10.1021/jm501124j},
journal = {Journal of Medicinal Chemistry},
number = 22,
volume = 57,
place = {United States},
year = {Fri Nov 07 00:00:00 EST 2014},
month = {Fri Nov 07 00:00:00 EST 2014}
}
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https://doi.org/10.1021/jm501124j
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