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U.S. Department of Energy
Office of Scientific and Technical Information

Applications of SFC-MS to toxins and compounds of biological interest

Conference ·
OSTI ID:7007067

The principal applications of supercritical fluid chromatography (SFC) are for compounds that are thermally labile, of low volatility, and of low to moderate polarity. Many compounds of biological and pharmaceutical interest are defined by these criteria. We have examined selected compounds of moderate to high molecular weight with biological activity. We have used the HFR interface with CO/sub 2/ as the mobile phase with from 2 to 5% modifier. One class of compounds potentially addressable by SFC-MS are cyclic peptides. These polar compounds require the use of polar fluid modifiers with CO/sub 2/ as the mobile phase. The ionic nature of the more hydrophilic portions of such polypeptides can sometimes be shielded, allowing solvation in supercritical fluid solvents. Cyclosporin A was successfully separated by SFC-MS using a microbore column using a 2% methanol modifier. The compound was also successfully separated with a capillary column. With the capillary column 2% 2-propanol was adequate, whereas with the microbore column more polar methanol was needed. The mass spectra were identical in both cases. We also analyzed the sodium salt of two ionic polyethers, digitoxigenin, digoxigenin, and cymarin. Results are briefly discussed. 5 refs.

Research Organization:
Pacific Northwest Lab., Richland, WA (USA)
DOE Contract Number:
AC06-76RL01830
OSTI ID:
7007067
Report Number(s):
PNL-SA-15741; CONF-8806199-3; ON: DE88014768
Country of Publication:
United States
Language:
English