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Halogenated pyrimidines as radiosensitizers for high-LET radiation

Journal Article · · Radiat. Res.; (United States)
DOI:https://doi.org/10.2307/3577336· OSTI ID:6276412
The incorporation of iododeoxyuridine (IdUrd) into Chinese hamster cells was examined as a possible radiosensitizer for fission spectrum neutrons. Dose-response curves comparing both X rays and neutrons in the same cell line with the same IdUrd replacement showed a similar radiation enhancement for IdUrd incorporation. Enhancement ratios at the 1% survival level were 1.8 for X rays and 1.5 for fission spectrum neutrons. While the mechanism of this enhancement in the response for fission neutron radiation is unclear, these positive data should support further exploration to determine if halogenated pyrimidine incorporation results in sensitization for neutron energies employed in therapy.
Research Organization:
National Cancer Institute, Bethesda, MD (USA)
OSTI ID:
6276412
Journal Information:
Radiat. Res.; (United States), Journal Name: Radiat. Res.; (United States) Vol. 117:2; ISSN RAREA
Country of Publication:
United States
Language:
English