Bivalent BET Bromodomain Inhibitors Confer Increased Potency and Selectivity for BRDT via Protein Co

Guan, Xianghong; Cheryala, Narsihmulu; Karim, Rezaul Md.; Chan, Alice; Berndt, Norbert; Qi, Jun; Georg, Gunda I.; Schonbrunn, Ernst

doi:10.1021/acs.jmedchem.2c00453

Bivalent BET Bromodomain Inhibitors Confer Increased Potency and Selectivity for BRDT via Protein Co

Journal Article · 01 July 2022 · J. Med. Chem.

DOI:https://doi.org/10.1021/acs.jmedchem.2c00453· OSTI ID:1901323

Guan, Xianghong; Cheryala, Narsihmulu; Karim, Rezaul Md.; Chan, Alice; Berndt, Norbert; Qi, Jun; Georg, Gunda I.; Schonbrunn, Ernst

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: DOE - Office Of Science; NCI

OSTI ID:: 1901323

Journal Information:: J. Med. Chem., Journal Name: J. Med. Chem. Journal Issue: (15) Vol. 65

Country of Publication:: United States

Language:: ENGLISH

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