Methylpyrrole inhibitors of BET bromodomains

Hasvold, Lisa A.; Sheppard, George S.; Wang, Le; Fidanze, Steven D.; Liu, Dachun; Pratt, John K.; Mantei, Robert A.; Wada, Carol K.; Hubbard, Robbert; Shen, Yu; Lin, Xiaoyu; Huang, Xiaoli; Warder, Scott E.; Wilcox, Denise; Li, Leiming; Buchanan, F. Greg; Smithee, Lauren; Albert, Daniel H.; Magoc, Terrance J.; Park, Chang H.; Petros, Andrew M.; Panchal, Sanjay C.; Sun, Chaohong; Kovar, Peter; Soni, Nirupama B.; Elmore, Steven W.; Kati, Warren M.; McDaniel, Keith F.

doi:10.1016/j.bmcl.2017.02.057

Methylpyrrole inhibitors of BET bromodomains

Journal Article · Mon May 01 00:00:00 EDT 2017 · Bioorganic and Medicinal Chemistry Letters

DOI:https://doi.org/10.1016/j.bmcl.2017.02.057· OSTI ID:1414004

Hasvold, Lisa A.; Sheppard, George S.; Wang, Le; Fidanze, Steven D.; Liu, Dachun; Pratt, John K.; Mantei, Robert A.; Wada, Carol K.; Hubbard, Robbert; Shen, Yu; Lin, Xiaoyu; Huang, Xiaoli; Warder, Scott E.; Wilcox, Denise; Li, Leiming; Buchanan, F. Greg; Smithee, Lauren; Albert, Daniel H.; Magoc, Terrance J.; Park, Chang H. more »

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View Accepted Manuscript (Publisher)

Sponsoring Organization:: USDOE

Grant/Contract Number:: AC02-06CH11357

OSTI ID:: 1414004

Alternate ID(s):: OSTI ID: 1400313

Journal Information:: Bioorganic and Medicinal Chemistry Letters, Journal Name: Bioorganic and Medicinal Chemistry Letters Journal Issue: 10 Vol. 27; ISSN 0960-894X

Publisher:: ElsevierCopyright Statement

Country of Publication:: United Kingdom

Language:: English

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Genome-wide siRNA screen identifies SMCX, EP400, and Brd4 as E2-dependent regulators of human papillomavirus oncogene expression Smith, Jennifer A.; White, Elizabeth A.; Sowa, Mathew E. Proceedings of the National Academy of Sciences, Vol. 107, Issue 8 https://doi.org/10.1073/pnas.0914818107	journal	February 2010
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