Discovery of acyl ureas as highly selective small molecule CSF1R kinase inhibitors

Caldwell, Timothy M.; Kaufman, Michael D.; Wise, Scott C.; Ahn, Yu Mi; Hood, Molly M.; Lu, Wei-Ping; Patt, William C.; Samarakoon, Thiwanka; Vogeti, Lakshminarayana; Vogeti, Subha; Yates, Karen M.; Bulfer, Stacie L.; Le Bourdonnec, Bertrand; Smith, Bryan D.; Flynn, Daniel L.

doi:10.1016/j.bmcl.2022.128929

Discovery of acyl ureas as highly selective small molecule CSF1R kinase inhibitors

Journal Article · Sat Oct 01 00:00:00 EDT 2022 · Bioorg. Med. Chem. Lett.

DOI:https://doi.org/10.1016/j.bmcl.2022.128929· OSTI ID:1900946

Caldwell, Timothy M.; Kaufman, Michael D.; Wise, Scott C.; Ahn, Yu Mi; Hood, Molly M.; Lu, Wei-Ping; Patt, William C.; Samarakoon, Thiwanka; Vogeti, Lakshminarayana; Vogeti, Subha; Yates, Karen M.; Bulfer, Stacie L.; Le Bourdonnec, Bertrand; Smith, Bryan D.; Flynn, Daniel L.

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: DOE - Office Of Science; INDUSTRY

OSTI ID:: 1900946

Journal Information:: Bioorg. Med. Chem. Lett., Journal Name: Bioorg. Med. Chem. Lett. Vol. 74

Country of Publication:: United States

Language:: ENGLISH

References (20)

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Discovery of acyl ureas as highly selective small molecule CSF1R kinase inhibitors

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