Development of LM98, a Small-Molecule TEAD Inhibitor Derived from Flufenamic Acid

Melin, Lea; Abdullayev, Shuay; Fnaiche, Ahmed; Vu, Victoria; Suarez, Narjara Gonzalez; Zeng, Hong; Szewczyk, Magdalena M.; Li, Fengling; Senisterra, Guillermo; Allali-Hassani, Abdellah; Chau, Irene; Dong, Aiping; Woo, Simon; Annabi, Borhane; Halabelian, Levon; LaPlante, Steven R.; Vedadi, Masoud; Barsyte-Lovejoy, Dalia; Santhakumar, Vijayaratnam; Gagnon, Alexandre

doi:10.1002/cmdc.202100432

Development of LM98, a Small-Molecule TEAD Inhibitor Derived from Flufenamic Acid

Journal Article · Fri Oct 01 00:00:00 EDT 2021 · ChemMedChem

DOI:https://doi.org/10.1002/cmdc.202100432· OSTI ID:1831264

Melin, Lea; Abdullayev, Shuay; Fnaiche, Ahmed; Vu, Victoria; Suarez, Narjara Gonzalez; Zeng, Hong; Szewczyk, Magdalena M.; Li, Fengling; Senisterra, Guillermo; Allali-Hassani, Abdellah; Chau, Irene; Dong, Aiping; Woo, Simon; Annabi, Borhane; Halabelian, Levon; LaPlante, Steven R.; Vedadi, Masoud; Barsyte-Lovejoy, Dalia; Santhakumar, Vijayaratnam; Gagnon, Alexandre

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: DOE - Office Of Science; FOREIGN; NIH

OSTI ID:: 1831264

Journal Information:: ChemMedChem, Journal Name: ChemMedChem Journal Issue: (19) Vol. 16

Country of Publication:: United States

Language:: ENGLISH

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