Development of Dimethylisoxazole-Attached Imidazo[1,2-a]pyridines as Potent and Selective CBP/P300 I

Muthengi, Alex; Wimalasena, Virangika K.; Yosief, Hailemichael O.; Bikowitz, Melissa J.; Sigua, Logan H.; Wang, Tingjian; Li, Deyao; Gaieb, Zied; Dhawan, Gagan; Liu, Shuai; Erickson, Jon; Amaro, Rommie E.; Schonbrunn, Ernst; Qi, Jun; Zhang, Wei

doi:10.1021/acs.jmedchem.0c02232

Development of Dimethylisoxazole-Attached Imidazo[1,2-a]pyridines as Potent and Selective CBP/P300 I

Journal Article · 01 April 2021 · J. Med. Chem.

DOI:https://doi.org/10.1021/acs.jmedchem.0c02232· OSTI ID:1787774

Muthengi, Alex; Wimalasena, Virangika K.; Yosief, Hailemichael O.; Bikowitz, Melissa J.; Sigua, Logan H.; Wang, Tingjian; Li, Deyao; Gaieb, Zied; Dhawan, Gagan; Liu, Shuai; Erickson, Jon; Amaro, Rommie E.; Schonbrunn, Ernst; Qi, Jun; Zhang, Wei

Research Organization:: Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Organization:: DOE - Office Of Science; NCI; National Institutes of Health (NIH)

OSTI ID:: 1787774

Journal Information:: J. Med. Chem., Vol. 64, Issue (9)

Country of Publication:: United States

Language:: ENGLISH

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