Characterization of novel small-molecule NRF2 activators: Structural and biochemical validation of stereospecific KEAP1 binding
Journal Article
·
· Biochimica et Biophysica Acta - General Subjects
Abstract not provided
- Research Organization:
- Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)
- Sponsoring Organization:
- INDUSTRY
- OSTI ID:
- 1347780
- Journal Information:
- Biochimica et Biophysica Acta - General Subjects, Journal Name: Biochimica et Biophysica Acta - General Subjects Journal Issue: 11 Vol. 1860; ISSN 0304-4165
- Publisher:
- Elsevier
- Country of Publication:
- United States
- Language:
- ENGLISH
Similar Records
Characterization of novel small-molecule NRF2 activators: Structural and biochemical validation of stereospecific KEAP1 binding
Small molecules inhibit the interaction of Nrf2 and the Keap1 Kelch domain through a non-covalent mechanism
Synthesis and Evaluation of Noncovalent Naphthalene-Based KEAP1-NRF2 Inhibitors
Journal Article
·
Mon Oct 31 20:00:00 EDT 2016
· Biochimica et Biophysica Acta - General Subjects
·
OSTI ID:1396468
Small molecules inhibit the interaction of Nrf2 and the Keap1 Kelch domain through a non-covalent mechanism
Journal Article
·
Tue Jul 30 00:00:00 EDT 2013
· Bioorgan. Med. Chem.
·
OSTI ID:1087768
Synthesis and Evaluation of Noncovalent Naphthalene-Based KEAP1-NRF2 Inhibitors
Journal Article
·
Tue Sep 01 00:00:00 EDT 2020
· ACS Medicinal Chemistry Letters
·
OSTI ID:1657586