Skip to main content
OSTI.GOVU.S. Department of Energy Office of Scientific and Technical Information
U.S. Department of Energy
Office of Scientific and Technical Information
 

Discovery of Benzotriazolo[4,3-d][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains

Journal Article · · ACS Med. Chem. Lett.
DOI:https://doi.org/10.1021/ml500411h· OSTI ID:1245844
; ; ; ; ; ; ; ; ; ; ; ; ; ; ; ; ; ; ; more »; ; ;  [1] « less
  1. Constellation
+ Show Author Affiliations
Abstract not provided
Research Organization:
Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)
Sponsoring Organization:
INDUSTRY
OSTI ID:
1245844
Journal Information:
ACS Med. Chem. Lett., Journal Name: ACS Med. Chem. Lett. Journal Issue: (2) ; 02, 2016 Vol. 7; ISSN 1948-5875
Country of Publication:
United States
Language:
ENGLISH

Similar Records

Structure-Based Discovery of CF53 as a Potent and Orally Bioavailable Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitor
Journal Article · Sat Jun 16 20:00:00 EDT 2018 · Journal of Medicinal Chemistry · OSTI ID:1471643
Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Usi
Journal Article · Wed Sep 01 00:00:00 EDT 2021 · J. Med. Chem. · OSTI ID:1832563
Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Usi
Journal Article · Wed Sep 01 00:00:00 EDT 2021 · J. Med. Chem. · OSTI ID:1834907

Related Subjects