Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors

Gehling, Victor S.; Hewitt, Michael C.; Vaswani, Rishi G.; Leblanc, Yves; Côté, Alexandre; Nasveschuk, Christopher G.; Taylor, Alexander M.; Harmange, Jean-Christophe; Audia, James E.; Pardo, Eneida; Joshi, Shivangi; Sandy, Peter; Mertz, Jennifer A.; Bergeron, Louise; Bryant, Barbara M.; Bellon, Steve; Poy, Florence; Jayaram, Hariharan; Sankaranarayanan, Ravichandran; Yellapantula, Sreegouri; Srinivasamurthy, Nandana Bangalore; Birudukota, Swarnakumari; Albrecht, Brian K.

doi:10.1021/ml4001485

Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors

Journal Article · Mon Oct 07 04:00:00 EDT 2013 · ACS Med. Chem. Lett.

DOI:https://doi.org/10.1021/ml4001485· OSTI ID:1095375

Gehling, Victor S.; Hewitt, Michael C.; Vaswani, Rishi G.; Leblanc, Yves; Côté, Alexandre; Nasveschuk, Christopher G.; Taylor, Alexander M.; Harmange, Jean-Christophe; Audia, James E.; Pardo, Eneida; Joshi, Shivangi; Sandy, Peter; Mertz, Jennifer A.; Bergeron, Louise; Bryant, Barbara M.; Bellon, Steve; Poy, Florence; Jayaram, Hariharan; Sankaranarayanan, Ravichandran; Yellapantula, Sreegouri more »

Jubilant

Abstract not provided

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: INDUSTRY

OSTI ID:: 1095375

Journal Information:: ACS Med. Chem. Lett., Journal Name: ACS Med. Chem. Lett. Journal Issue: (9) ; 09, 2013 Vol. 4

Country of Publication:: United States

Language:: ENGLISH

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Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors

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