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9-{beta}-arabinofuranosyladenine preferentially sensitizes radioresistant squamous cell carcinoma cell lines to x-rays

Technical Report ·
DOI:https://doi.org/10.2172/10149645· OSTI ID:10149645
 [1];  [2];  [2]
  1. Rush Univ. Medical Center, Chicago, IL (United States). Therapeutic Radiology
  2. Chicago Univ., IL (United States). Dept. of Radiation and Cellular Oncology
The effect of 9-{beta}-arabinofuranosyladenine (ara-A) on sensitivity to the deleterious effects of x-rays was studied in six squamous cell carcinoma cell lines. Three lines were relatively radioresistant, having D{sub 0} values of 2.31 to 2.89 Gy, and the other three lines were relatively radiosensitive, having D{sub 0} values of between 1.07 and 1.45 Gy. Ara-A (50 or 500 {mu}M) was added to cultures 30 min prior to irradiation and removed 30 min after irradiation, and sensitivity was measured in terms of cell survival. The radiosensitizing effect of ara-A was very dependent on the inherent radiosensitivity of the tumor cell line. Fifty micromolar concentrations of ara-A sensitized only the two most radioresistant lines, SCC-12B.2 and JSQ-3. Five hundred micromolar concentrations of ara-A sensitized the more sensitive cell lines, SQ-20B and SQ-9G, but failed to have any effect on the radiation response of the two most sensitive cell lines, SQ-38 and SCC-61. Concentrations of ara-A as low as 10 {mu}M were equally efficient in inhibiting DNA synthesis in all six cell lines. These results suggest that the target for the radiosensitizing effect of ara-A is probably related to the factor controlling the inherent radiosensitivity of human tumor cells. Therefore, ara-A might be useful in overcoming radiation resistance in vivo.
Research Organization:
Argonne National Lab., IL (United States); Chicago Univ., IL (United States). Dept. of Radiation and Cellular Oncology
Sponsoring Organization:
USDOE, Washington, DC (United States); National Cancer Inst., Bethesda, MD (United States)
DOE Contract Number:
W-31109-ENG-38; FG02-88ER60661
OSTI ID:
10149645
Report Number(s):
ANL/BIM/PP--76541; ON: DE94011510; BR: HA0202010; CNN: CA 42596
Country of Publication:
United States
Language:
English

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