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Title: From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors

Authors:
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Publication Date:
Type:
Publisher's Accepted Manuscript
Journal Name:
Bioorganic and Medicinal Chemistry Letters
Additional Journal Information:
Journal Name: Bioorganic and Medicinal Chemistry Letters Journal Volume: 27 Journal Issue: 13; Journal ID: ISSN 0960-894X
Publisher:
Elsevier
Sponsoring Org:
USDOE
Country of Publication:
United Kingdom
Language:
English
OSTI Identifier:
1413842

Liang, Jun, Labadie, Sharada, Zhang, Birong, Ortwine, Daniel F., Patel, Snahel, Vinogradova, Maia, Kiefer, James R., Mauer, Till, Gehling, Victor S., Harmange, Jean-Christophe, Cummings, Richard, Lai, Tommy, Liao, Jiangpeng, Zheng, Xiaoping, Liu, Yichin, Gustafson, Amy, Van der Porten, Erica, Mao, Weifeng, Liederer, Bianca M., Deshmukh, Gauri, An, Le, Ran, Yingqing, Classon, Marie, Trojer, Patrick, Dragovich, Peter S., and Murray, Lesley. From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors. United Kingdom: N. p., Web. doi:10.1016/j.bmcl.2017.05.016.
Liang, Jun, Labadie, Sharada, Zhang, Birong, Ortwine, Daniel F., Patel, Snahel, Vinogradova, Maia, Kiefer, James R., Mauer, Till, Gehling, Victor S., Harmange, Jean-Christophe, Cummings, Richard, Lai, Tommy, Liao, Jiangpeng, Zheng, Xiaoping, Liu, Yichin, Gustafson, Amy, Van der Porten, Erica, Mao, Weifeng, Liederer, Bianca M., Deshmukh, Gauri, An, Le, Ran, Yingqing, Classon, Marie, Trojer, Patrick, Dragovich, Peter S., & Murray, Lesley. From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors. United Kingdom. doi:10.1016/j.bmcl.2017.05.016.
Liang, Jun, Labadie, Sharada, Zhang, Birong, Ortwine, Daniel F., Patel, Snahel, Vinogradova, Maia, Kiefer, James R., Mauer, Till, Gehling, Victor S., Harmange, Jean-Christophe, Cummings, Richard, Lai, Tommy, Liao, Jiangpeng, Zheng, Xiaoping, Liu, Yichin, Gustafson, Amy, Van der Porten, Erica, Mao, Weifeng, Liederer, Bianca M., Deshmukh, Gauri, An, Le, Ran, Yingqing, Classon, Marie, Trojer, Patrick, Dragovich, Peter S., and Murray, Lesley. 2017. "From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors". United Kingdom. doi:10.1016/j.bmcl.2017.05.016.
@article{osti_1413842,
title = {From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors},
author = {Liang, Jun and Labadie, Sharada and Zhang, Birong and Ortwine, Daniel F. and Patel, Snahel and Vinogradova, Maia and Kiefer, James R. and Mauer, Till and Gehling, Victor S. and Harmange, Jean-Christophe and Cummings, Richard and Lai, Tommy and Liao, Jiangpeng and Zheng, Xiaoping and Liu, Yichin and Gustafson, Amy and Van der Porten, Erica and Mao, Weifeng and Liederer, Bianca M. and Deshmukh, Gauri and An, Le and Ran, Yingqing and Classon, Marie and Trojer, Patrick and Dragovich, Peter S. and Murray, Lesley},
abstractNote = {},
doi = {10.1016/j.bmcl.2017.05.016},
journal = {Bioorganic and Medicinal Chemistry Letters},
number = 13,
volume = 27,
place = {United Kingdom},
year = {2017},
month = {7}
}