Skip to main content
U.S. Department of Energy
Office of Scientific and Technical Information

Models for bacteriorhodopsin-catalyzed dark cis-trans isomerization of bound retinal

Journal Article · · Journal of the American Chemical Society; (USA)
DOI:https://doi.org/10.1021/ja00167a054· OSTI ID:6649597
 [1]
  1. Brookhaven National Laboratory, Upton, NY (USA)

The syntheses of syn- and anti-2-aza-6-carboxymethylbicyclo(2.2.2)octane and syn and anti-2-aza-6-carboxypropyl(2.2.2)octane zwitterions are described. These compounds, which have secondary amines to form positively charged Schiff bases with retinal and a pendant carboxylate anion to interact with the polyeniminium system, mimic the presence of aspartate-212 and lysine-216 at the retinal binding/cis-trans isomerization site of bacteriorhodopsin. Kinetics of retinal cis-trans isomerization of these model compounds are reported and are discussed in light of previous MNDO calculations (J. Am. Chem. Soc. 1987, 109, 1627-1631) of isomerization barrier heights affected by the movement of an anion to different positions with respect to the polyeniminium system.

DOE Contract Number:
AC02-76CH00016
OSTI ID:
6649597
Journal Information:
Journal of the American Chemical Society; (USA), Journal Name: Journal of the American Chemical Society; (USA) Vol. 112:11; ISSN 0002-7863; ISSN JACSA
Country of Publication:
United States
Language:
English