Defining the structure-activity relationship for a novel class of allosteric MKP5 inhibitors

Gannam, Zachary T.K.; Jamali, Haya; Kweon, Oh Sang; Herrington, James; Shillingford, Shanelle R.; Papini, Christina; Gentzel, Erik; Lolis, Elias; Bennett, Anton M.; Ellman, Jonathan A.; Anderson, Karen S.

doi:10.1016/j.ejmech.2022.114712

Defining the structure-activity relationship for a novel class of allosteric MKP5 inhibitors

Journal Article · 30 November 2022 · Eur. J. Med. Chem.

DOI:https://doi.org/10.1016/j.ejmech.2022.114712· OSTI ID:1901313

Gannam, Zachary T.K.; Jamali, Haya; Kweon, Oh Sang; Herrington, James; Shillingford, Shanelle R.; Papini, Christina; Gentzel, Erik; Lolis, Elias; Bennett, Anton M.; Ellman, Jonathan A.; Anderson, Karen S.

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: DOE - Office Of Science; NIH

OSTI ID:: 1901313

Journal Information:: Eur. J. Med. Chem., Journal Name: Eur. J. Med. Chem. Vol. 243

Country of Publication:: United States

Language:: ENGLISH

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