Defining the structure-activity relationship for a novel class of allosteric MKP5 inhibitors

Gannam, Zachary T.K.; Jamali, Haya; Kweon, Oh Sang; Herrington, James; Shillingford, Shanelle R.; Papini, Christina; Gentzel, Erik; Lolis, Elias; Bennett, Anton M.; Ellman, Jonathan A.; Anderson, Karen S.

doi:10.1016/j.ejmech.2022.114712

Title: Defining the structure-activity relationship for a novel class of allosteric MKP5 inhibitors

Journal Article · 01 December 2022 · Eur. J. Med. Chem.

DOI:https://doi.org/10.1016/j.ejmech.2022.114712· OSTI ID:1901313

Gannam, Zachary T.K.; Jamali, Haya; Kweon, Oh Sang; Herrington, James; Shillingford, Shanelle R.; Papini, Christina; Gentzel, Erik; Lolis, Elias; Bennett, Anton M.; Ellman, Jonathan A.; Anderson, Karen S.

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Research Organization:: Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Organization:: DOE - Office Of Science; National Institutes of Health (NIH)

OSTI ID:: 1901313

Journal Information:: Eur. J. Med. Chem., Vol. 243

Country of Publication:: United States

Language:: ENGLISH

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