Discovery and Optimization of Highly Selective Inhibitors of CDK5

Daniels, Matthew H.; Malojcic, Goran; Clugston, Susan L.; Williams, Brett; Gal, Marie Coeffet-Le; Pan-Zhou, Xin-Ru; Venkatachalan, Srinivasan; Harmange, Jean-Christophe; Ledeboer, Mark

doi:10.1021/acs.jmedchem.1c02069

Discovery and Optimization of Highly Selective Inhibitors of CDK5

Journal Article · 31 January 2022 · J. Med. Chem.

DOI:https://doi.org/10.1021/acs.jmedchem.1c02069· OSTI ID:1865460

Daniels, Matthew H.; Malojcic, Goran; Clugston, Susan L.; Williams, Brett; Gal, Marie Coeffet-Le; Pan-Zhou, Xin-Ru; Venkatachalan, Srinivasan; Harmange, Jean-Christophe; Ledeboer, Mark

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: DOE - Office Of Science; INDUSTRY

OSTI ID:: 1865460

Journal Information:: J. Med. Chem., Journal Name: J. Med. Chem. Journal Issue: (4) Vol. 65

Country of Publication:: United States

Language:: ENGLISH

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