Preparation and biological evaluation of conformationally constrained BACE1 inhibitors

Winneroski, Leonard L.; Schiffler, Matthew A.; Erickson, Jon A.; May, Patrick C.; Monk, Scott A.; Timm, David E.; Audia, James E.; Beck, James P.; Boggs, Leonard N.; Borders, Anthony R.; Boyer, Robert D.; Brier, Richard A.; Hudziak, Kevin J.; Klimkowski, Valentine J.; Losada, Pablo Garcia; Mathes, Brian M.; Stout, Stephanie L.; Watson, Brian M.; Mergott, Dustin J.

doi:10.1016/j.bmc.2015.04.062

Preparation and biological evaluation of conformationally constrained BACE1 inhibitors

Journal Article · Wed Jul 01 04:00:00 EDT 2015 · Bioorgan. Med. Chem.

DOI:https://doi.org/10.1016/j.bmc.2015.04.062· OSTI ID:1856369

Winneroski, Leonard L.; Schiffler, Matthew A.; Erickson, Jon A.; May, Patrick C.; Monk, Scott A.; Timm, David E.; Audia, James E.; Beck, James P.; Boggs, Leonard N.; Borders, Anthony R.; Boyer, Robert D.; Brier, Richard A.; Hudziak, Kevin J.; Klimkowski, Valentine J.; Losada, Pablo Garcia; Mathes, Brian M.; Stout, Stephanie L.; Watson, Brian M.; Mergott, Dustin J.

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: DOE - Office Of Science; INDUSTRY

OSTI ID:: 1856369

Journal Information:: Bioorgan. Med. Chem., Journal Name: Bioorgan. Med. Chem. Journal Issue: (13) Vol. 23

Country of Publication:: United States

Language:: ENGLISH

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