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Transformation of Carbonyl Compounds into Homologous Alkynes under Neutral Conditions: Fragmentation of Tetrazoles Derived from Cyanophosphates
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journal
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May 2017 |
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Synthesis of Spirocyclic Pyrrolidines: Advanced Building Blocks for Drug Discovery
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journal
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October 2017 |
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Total syntheses of the squalene-derived halogenated polyethers ent -dioxepandehydrothyrsiferol and armatol A via bromonium- and Lewis acid-initiated epoxide-opening cascades
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June 2013 |
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Discovery and Optimization of Rationally Designed Bicyclic Inhibitors of Human Arginase to Enhance Cancer Immunotherapy
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March 2020 |
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Discovery of ( R )-2-Amino-6-borono-2-(2-(piperidin-1-yl)ethyl)hexanoic Acid and Congeners As Highly Potent Inhibitors of Human Arginases I and II for Treatment of Myocardial Reperfusion Injury
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journal
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March 2013 |
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Collagen Stability: Insights from NMR Spectroscopic and Hybrid Density Functional Computational Investigations of the Effect of Electronegative Substituents on Prolyl Ring Conformations
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journal
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February 2002 |
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Bicyclic proline analogues as organocatalysts for stereoselective aldol reactions: an in silico DFT study
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January 2007 |
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The importance of synthetic chemistry in the pharmaceutical industry
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journal
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January 2019 |
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Synthesis and Anti-HIV Activity of d - and l -Thietanose Nucleosides
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journal
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February 2006 |
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A new method of synthesis of methyl N-Boc-2,3-dehydropyrrolidine- and piperidine-2-carboxylates
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journal
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June 2008 |
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trans-3-n-propyl-L-proline is a highly favorable, conformationally restricted replacement for methionine in the C-terminal tetrapeptide of cholecystokinin. Stereoselective synthesis of 3-allyl- and 3-n-propyl-L-proline derivatives from 4-hydroxy-L-proline
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January 1991 |
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Collagen Structure and Stability
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June 2009 |
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Escaping from Flatland: Antimalarial Activity of sp 3 -Rich Bridged Pyrrolidine Derivatives
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November 2020 |
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Influence of proline residues on protein conformation
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March 1991 |
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Finding the Perfect Match: A Combined Computational and Experimental Study toward Efficient and Scalable Photosensitized [2 + 2] Cycloadditions in Flow
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journal
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December 2018 |
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[2+2] Cycloaddition reaction of cyclic enecarbamates and enamides with ketenes. A short and efficient synthesis of the Geissman-Waiss lactone.
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journal
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January 1993 |
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A scalable synthesis of (1R,3S,5R)-2-(tert-butoxycarbonyl)-2-azabicyclo[3.1.0]hexane-3-carboxylic acid
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journal
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December 2013 |
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Synthesis of Chiral Tetrahydrofuran Building Blocks from Pantolactones: Application in the Synthesis of Empagliflozin and Amprenavir Analogs: Synthesis of Chiral Tetrahydrofuran Building Blocks from Pantolactones: Application in the Synthesis of Empagliflozin and Amprenavir Analogs
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journal
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July 2019 |
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L-arginine metabolism in myeloid cells controls T-lymphocyte functions
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journal
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June 2003 |
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Synthesis of [ c ]-Fused Bicyclic Proline Analogues: Synthesis of [ c ]-Fused Bicyclic Proline Analogues
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journal
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January 2015 |
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A new method for the deoxygenation of secondary alcohols
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journal
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January 1975 |
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Synthesis and properties of pinanediol .alpha.-amido boronic esters
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journal
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August 1984 |
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Synthesis of Bicyclic Proline Derivatives by the Aza-Cope-Mannich Reaction: Formal Synthesis of (±)-Acetylaranotin
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journal
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January 2015 |
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A novel approach to 2,4-ethanoproline
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journal
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July 2009 |
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Asymmetric construction of benzylic quaternary carbons from chiral malonates: Formal synthesis of natural (−)aphanorphine
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journal
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April 1995 |
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Correlations between catalytic reactions of diazo compounds and stoichiometric reactions of transition-metal carbenes with alkenes. Mechanism of the cyclopropanation reaction
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journal
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January 1984 |
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A Spectrophotometric Assay of Arginase
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journal
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August 2001 |
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Enantiospecific Synthesis of Heterocycles from α-Amino Acids
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journal
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January 1996 |
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Use of hexamethylphosphoramide chmpa in the alkylation of aromatic amines: synthesis of azetidines, pyrrolidines, piperidines and hexahydroazepines
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journal
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January 1989 |
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Asymmetric synthesis of S-(−)-cucurbitine
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journal
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November 1992 |
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Development of a Zinc-Mediated Approach to a 2,3- cis -Pyrrolidine Arginase Inhibitor
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journal
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June 2020 |
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A Convenient Two-Step Procedure for the Synthesis of Substituted Allylic Amines from Allylic Alcohols
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journal
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July 1995 |
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Discovery of N -Substituted 3-Amino-4-(3-boronopropyl)pyrrolidine-3-carboxylic Acids as Highly Potent Third-Generation Inhibitors of Human Arginase I and II
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journal
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August 2019 |
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Structure-Based Discovery of Proline-Derived Arginase Inhibitors with Improved Oral Bioavailability for Immuno-Oncology
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journal
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July 2021 |
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Iridium-catalyzed hydroboration of alkenes with pinacolborane
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journal
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November 2004 |
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Inhibition of arginase by CB-1158 blocks myeloid cell-mediated immune suppression in the tumor microenvironment
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journal
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December 2017 |
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Organic synthesis provides opportunities to transform drug discovery
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journal
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March 2018 |
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Synthesis of Cyclobutane-Fused Angular Tetracyclic Spiroindolines via Visible-Light-Promoted Intramolecular Dearomatization of Indole Derivatives
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journal
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January 2019 |
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A Medicinal Chemist’s Guide to Molecular Interactions
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journal
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July 2010 |
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Regulation of arginase I activity and expression by both PD-1 and CTLA-4 on the myeloid-derived suppressor cells
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journal
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October 2008 |
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A Novel Class of Tunable Zinc Reagents (RXZnCH 2 Y) for Efficient Cyclopropanation of Olefins
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journal
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December 2003 |
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Synthetic Strategy toward the Pentacyclic Core of Melodinus Alkaloids
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journal
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January 2018 |
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Arginase Inhibitors: A Rational Approach Over One Century: AN EXHAUSTIVE REVIEW OF ARGINASE INHIBITORS
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journal
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November 2016 |
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The crystal structure of DL -proline hydrochloride
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journal
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November 1969 |
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Binding of α,α-Disubstituted Amino Acids to Arginase Suggests New Avenues for Inhibitor Design
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journal
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August 2011 |
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Responsive Mn(II) complexes for potential applications in diagnostic Magnetic Resonance Imaging
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journal
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February 2011 |
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Asymmetric Synthesis of Unsaturated, Fused Bicyclic Proline Analogues through Amino Alkylation of Cyclic Bis(allylsulfoximine)titanium Complexes and Migratory Cyclization of δ-Amino Alkenyl Aminosulfoxonium Salts
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journal
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October 2003 |
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Small Molecule Conformational Preferences Derived from Crystal Structure Data. A Medicinal Chemistry Focused Analysis
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journal
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December 2007 |
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Chiral, bicyclic proline derivatives and their application as ligands for copper in the catalytic asymmetric allylic oxidation of olefins
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journal
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October 1996 |
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Efficient method for inversion of secondary alcohols by reaction of chloromethanesulfonates with cesium acetate
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journal
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August 1996 |