]Discovery of AM-6494: A Potent and Orally Efficacious [beta]-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitor with in Vivo Selectivity over BACE2
- Amgen
Abstract not provided
- Research Organization:
- Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)
- Sponsoring Organization:
- INDUSTRY
- OSTI ID:
- 1608844
- Journal Information:
- J. Med. Chem., Journal Name: J. Med. Chem. Journal Issue: (5) ; 01, 2020 Vol. 63
- Country of Publication:
- United States
- Language:
- ENGLISH
Similar Records
Discovery of furo[2,3-d][1,3]thiazinamines as beta amyloid cleaving enzyme-1 (BACE1) inhibitors
Discovery of potent iminoheterocycle BACE1 inhibitors
Design and Validation of Bicyclic Iminopyrimidinones As Beta Amyloid Cleaving Enzyme-1 (BACE1) Inhibitors: Conformational Constraint to Favor a Bioactive Conformation
Journal Article
·
Wed Nov 30 23:00:00 EST 2016
· Bioorganic & Medicinal Chemistry Letters
·
OSTI ID:1347755
Discovery of potent iminoheterocycle BACE1 inhibitors
Journal Article
·
Fri Sep 18 00:00:00 EDT 2015
· Bioorg. Med. Chem. Lett.
·
OSTI ID:1194208
Design and Validation of Bicyclic Iminopyrimidinones As Beta Amyloid Cleaving Enzyme-1 (BACE1) Inhibitors: Conformational Constraint to Favor a Bioactive Conformation
Journal Article
·
Tue Jun 11 00:00:00 EDT 2013
· J. Med. Chem.
·
OSTI ID:1083344