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Title: Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers

Authors:
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  1. Novartis
Publication Date:
Research Org.:
Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
Sponsoring Org.:
INDUSTRY
OSTI Identifier:
1545844
Resource Type:
Journal Article
Journal Name:
J. Med. Chem.
Additional Journal Information:
Journal Volume: 61; Journal Issue: (22) ; 11, 2018
Country of Publication:
United States
Language:
ENGLISH

Citation Formats

Papillon, Julien P.N., Nakajima, Katsumasa, Adair, Christopher D., Hempel, Jonathan, Jouk, Andriana O., Karki, Rajeshri G., Mathieu, Simon, Möbitz, Henrik, Ntaganda, Rukundo, Smith, Troy, Visser, Michael, Hill, Susan E., Hurtado, Felipe Kellermann, Chenail, Gregg, Bhang, Hyo-Eun C., Bric, Anka, Xiang, Kay, Bushold, Geoffrey, Gilbert, Tamara, Vattay, Anthony, Dooley, Julie, Costa, Emily A., Park, Isabel, Li, Ailing, Farley, David, Lounkine, Eugen, Yue, Q. Kimberley, Xie, Xiaoling, Zhu, Xiaoping, Kulathila, Raviraj, King, Daniel, Hu, Tiancen, Vulic, Katarina, Cantwell, John, Luu, Catherine, and Jagani, Zainab. Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers. United States: N. p., 2019. Web. doi:10.1021/acs.jmedchem.8b01318.
Papillon, Julien P.N., Nakajima, Katsumasa, Adair, Christopher D., Hempel, Jonathan, Jouk, Andriana O., Karki, Rajeshri G., Mathieu, Simon, Möbitz, Henrik, Ntaganda, Rukundo, Smith, Troy, Visser, Michael, Hill, Susan E., Hurtado, Felipe Kellermann, Chenail, Gregg, Bhang, Hyo-Eun C., Bric, Anka, Xiang, Kay, Bushold, Geoffrey, Gilbert, Tamara, Vattay, Anthony, Dooley, Julie, Costa, Emily A., Park, Isabel, Li, Ailing, Farley, David, Lounkine, Eugen, Yue, Q. Kimberley, Xie, Xiaoling, Zhu, Xiaoping, Kulathila, Raviraj, King, Daniel, Hu, Tiancen, Vulic, Katarina, Cantwell, John, Luu, Catherine, & Jagani, Zainab. Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers. United States. doi:10.1021/acs.jmedchem.8b01318.
Papillon, Julien P.N., Nakajima, Katsumasa, Adair, Christopher D., Hempel, Jonathan, Jouk, Andriana O., Karki, Rajeshri G., Mathieu, Simon, Möbitz, Henrik, Ntaganda, Rukundo, Smith, Troy, Visser, Michael, Hill, Susan E., Hurtado, Felipe Kellermann, Chenail, Gregg, Bhang, Hyo-Eun C., Bric, Anka, Xiang, Kay, Bushold, Geoffrey, Gilbert, Tamara, Vattay, Anthony, Dooley, Julie, Costa, Emily A., Park, Isabel, Li, Ailing, Farley, David, Lounkine, Eugen, Yue, Q. Kimberley, Xie, Xiaoling, Zhu, Xiaoping, Kulathila, Raviraj, King, Daniel, Hu, Tiancen, Vulic, Katarina, Cantwell, John, Luu, Catherine, and Jagani, Zainab. Fri . "Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers". United States. doi:10.1021/acs.jmedchem.8b01318.
@article{osti_1545844,
title = {Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers},
author = {Papillon, Julien P.N. and Nakajima, Katsumasa and Adair, Christopher D. and Hempel, Jonathan and Jouk, Andriana O. and Karki, Rajeshri G. and Mathieu, Simon and Möbitz, Henrik and Ntaganda, Rukundo and Smith, Troy and Visser, Michael and Hill, Susan E. and Hurtado, Felipe Kellermann and Chenail, Gregg and Bhang, Hyo-Eun C. and Bric, Anka and Xiang, Kay and Bushold, Geoffrey and Gilbert, Tamara and Vattay, Anthony and Dooley, Julie and Costa, Emily A. and Park, Isabel and Li, Ailing and Farley, David and Lounkine, Eugen and Yue, Q. Kimberley and Xie, Xiaoling and Zhu, Xiaoping and Kulathila, Raviraj and King, Daniel and Hu, Tiancen and Vulic, Katarina and Cantwell, John and Luu, Catherine and Jagani, Zainab},
abstractNote = {},
doi = {10.1021/acs.jmedchem.8b01318},
journal = {J. Med. Chem.},
number = (22) ; 11, 2018,
volume = 61,
place = {United States},
year = {2019},
month = {7}
}