R -Configuration of 4-Aminopyridyl-Based Inhibitors of CYP51 Confers Superior Efficacy Against Trypanosoma cruzi

Choi, Jun Yong; Calvet, Claudia M.; Vieira, Debora F.; Gunatilleke, Shamila S.; Cameron, Michael D.; McKerrow, James H.; Podust, Larissa M.; Roush, William R.

doi:10.1021/ml500010m

Title: R -Configuration of 4-Aminopyridyl-Based Inhibitors of CYP51 Confers Superior Efficacy Against Trypanosoma cruzi

Journal Article · Wed Jan 22 00:00:00 EST 2014 · ACS Medicinal Chemistry Letters

DOI:https://doi.org/10.1021/ml500010m· OSTI ID:1168423

Choi, Jun Yong ^[1]; Calvet, Claudia M. ^[2]; Vieira, Debora F.; Gunatilleke, Shamila S.; Cameron, Michael D. ^[3]; McKerrow, James H.; Podust, Larissa M.; Roush, William R. ^[1]

Department of Chemistry, Scripps Florida, Jupiter, Florida 33458, United States
Cellular Ultra-Structure Laboratory, Oswaldo Cruz Institute (IOC), FIOCRUZ, Rio de Janeiro, RJ 21040-362, Brazil
Department of Molecular Therapeutics, Scripps Florida, Jupiter, Florida 33458, United States

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Sponsoring Organization:: USDOE Office of Science (SC), Basic Energy Sciences (BES)

Grant/Contract Number:: AC02-05CH11231

OSTI ID:: 1168423

Journal Information:: ACS Medicinal Chemistry Letters, Journal Name: ACS Medicinal Chemistry Letters Vol. 5 Journal Issue: 4; ISSN 1948-5875

Publisher:: American Chemical SocietyCopyright Statement

Country of Publication:: United States

Language:: English

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Cited by: 19 works

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