Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV
- Authors:
-
- Yale Univ., New Haven, CT (United States)
- Publication Date:
- Research Org.:
- Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
- Sponsoring Org.:
- USDOE; National Institutes of Health (NIH)
- OSTI Identifier:
- 1547408
- Alternate Identifier(s):
- OSTI ID: 1636807
- Grant/Contract Number:
- AC02-06CH11357; AI044616; GM049551; AI141172; AI112443; AI122384; EB000487; S10OD021527; P30 GM124165
- Resource Type:
- Accepted Manuscript
- Journal Name:
- Antiviral Research
- Additional Journal Information:
- Journal Volume: 167; Journal Issue: 07, 2019; Journal ID: ISSN 0166-3542
- Publisher:
- Elsevier
- Country of Publication:
- United States
- Language:
- ENGLISH
- Subject:
- 60 APPLIED LIFE SCIENCES; HIV-1; non-nucleoside reverse transcriptase inhibitor; long-acting nanoformulation; pharmacokinetic studies; mice model; x-ray crystallography
Citation Formats
Kudalkar, Shalley N., Ullah, Irfan, Bertoletti, Nicole, Mandl, Hanna K., Cisneros, José A., Beloor, Jagadish, Chan, Albert H., Quijano, Elias, Saltzman, W. Mark, Jorgensen, William L., Kumar, Priti, and Anderson, Karen S. Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV. United States: N. p., 2019.
Web. doi:10.1016/j.antiviral.2019.04.010.
Kudalkar, Shalley N., Ullah, Irfan, Bertoletti, Nicole, Mandl, Hanna K., Cisneros, José A., Beloor, Jagadish, Chan, Albert H., Quijano, Elias, Saltzman, W. Mark, Jorgensen, William L., Kumar, Priti, & Anderson, Karen S. Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV. United States. https://doi.org/10.1016/j.antiviral.2019.04.010
Kudalkar, Shalley N., Ullah, Irfan, Bertoletti, Nicole, Mandl, Hanna K., Cisneros, José A., Beloor, Jagadish, Chan, Albert H., Quijano, Elias, Saltzman, W. Mark, Jorgensen, William L., Kumar, Priti, and Anderson, Karen S. Fri .
"Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV". United States. https://doi.org/10.1016/j.antiviral.2019.04.010. https://www.osti.gov/servlets/purl/1547408.
@article{osti_1547408,
title = {Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV},
author = {Kudalkar, Shalley N. and Ullah, Irfan and Bertoletti, Nicole and Mandl, Hanna K. and Cisneros, José A. and Beloor, Jagadish and Chan, Albert H. and Quijano, Elias and Saltzman, W. Mark and Jorgensen, William L. and Kumar, Priti and Anderson, Karen S.},
abstractNote = {},
doi = {10.1016/j.antiviral.2019.04.010},
journal = {Antiviral Research},
number = 07, 2019,
volume = 167,
place = {United States},
year = {Fri Apr 26 00:00:00 EDT 2019},
month = {Fri Apr 26 00:00:00 EDT 2019}
}
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Cited by: 12 works
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Works referencing / citing this record:
Structural insights into the recognition of nucleoside reverse transcriptase inhibitors by HIV‐1 reverse transcriptase: First crystal structures with reverse transcriptase and the active triphosphate forms of lamivudine and emtricitabine
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