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Title: Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging

Authors:
 [1];  [2];  [1];  [2];  [2];  [2];  [3];  [2];  [2];  [2];  [2];  [2];  [2];  [2];  [2];  [2];  [2];  [2];  [2];  [3] more »;  [2];  [1];  [1];  [1];  [4];  [5];  [6];  [5];  [4];  [1];  [2];  [1] « less
  1. Gordon Center for Medical Imaging & Nuclear Medicine and Molecular Imaging, Massachusetts General Hospital & Department of Radiology, Harvard Medical School, Boston MA 02114 USA
  2. Pfizer Worldwide Research and Development, Groton Laboratories, Eastern Point Road Groton CT 06340 USA
  3. Pfizer Worldwide Research and Development, 610 Main Street Cambridge MA 02139 USA
  4. Departments of Neurology & Psychiatry, Massachusetts General Hospital, Harvard Medical School, 185 Cambridge Street Boston MA 02114 USA
  5. Stanley Center for Psychiatric Research, Broad Institute, 415 Main Street Cambridge MA o2142 USA
  6. Stanley Center for Psychiatric Research, Broad Institute, 415 Main Street Cambridge MA o2142 USA, Departments of Neurology & Psychiatry, Massachusetts General Hospital, Harvard Medical School, 185 Cambridge Street Boston MA 02114 USA
Publication Date:
Sponsoring Org.:
USDOE
OSTI Identifier:
1400568
Grant/Contract Number:  
AC02-06CH11357
Resource Type:
Publisher's Accepted Manuscript
Journal Name:
Angewandte Chemie (International Edition)
Additional Journal Information:
Journal Name: Angewandte Chemie (International Edition) Journal Volume: 55 Journal Issue: 33; Journal ID: ISSN 1433-7851
Publisher:
Wiley Blackwell (John Wiley & Sons)
Country of Publication:
Germany
Language:
English

Citation Formats

Liang, Steven H., Chen, Jinshan Michael, Normandin, Marc D., Chang, Jeanne S., Chang, George C., Taylor, Christine K., Trapa, Patrick, Plummer, Mark S., Para, Kimberly S., Conn, Edward L., Lopresti-Morrow, Lori, Lanyon, Lorraine F., Cook, James M., Richter, Karl E. G., Nolan, Charlie E., Schachter, Joel B., Janat, Fouad, Che, Ye, Shanmugasundaram, Veerabahu, Lefker, Bruce A., Enerson, Bradley E., Livni, Elijahu, Wang, Lu, Guehl, Nicolas J., Patnaik, Debasis, Wagner, Florence F., Perlis, Roy, Holson, Edward B., Haggarty, Stephen J., El Fakhri, Georges, Kurumbail, Ravi G., and Vasdev, Neil. Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging. Germany: N. p., 2016. Web. doi:10.1002/anie.201603797.
Liang, Steven H., Chen, Jinshan Michael, Normandin, Marc D., Chang, Jeanne S., Chang, George C., Taylor, Christine K., Trapa, Patrick, Plummer, Mark S., Para, Kimberly S., Conn, Edward L., Lopresti-Morrow, Lori, Lanyon, Lorraine F., Cook, James M., Richter, Karl E. G., Nolan, Charlie E., Schachter, Joel B., Janat, Fouad, Che, Ye, Shanmugasundaram, Veerabahu, Lefker, Bruce A., Enerson, Bradley E., Livni, Elijahu, Wang, Lu, Guehl, Nicolas J., Patnaik, Debasis, Wagner, Florence F., Perlis, Roy, Holson, Edward B., Haggarty, Stephen J., El Fakhri, Georges, Kurumbail, Ravi G., & Vasdev, Neil. Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging. Germany. doi:10.1002/anie.201603797.
Liang, Steven H., Chen, Jinshan Michael, Normandin, Marc D., Chang, Jeanne S., Chang, George C., Taylor, Christine K., Trapa, Patrick, Plummer, Mark S., Para, Kimberly S., Conn, Edward L., Lopresti-Morrow, Lori, Lanyon, Lorraine F., Cook, James M., Richter, Karl E. G., Nolan, Charlie E., Schachter, Joel B., Janat, Fouad, Che, Ye, Shanmugasundaram, Veerabahu, Lefker, Bruce A., Enerson, Bradley E., Livni, Elijahu, Wang, Lu, Guehl, Nicolas J., Patnaik, Debasis, Wagner, Florence F., Perlis, Roy, Holson, Edward B., Haggarty, Stephen J., El Fakhri, Georges, Kurumbail, Ravi G., and Vasdev, Neil. Wed . "Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging". Germany. doi:10.1002/anie.201603797.
@article{osti_1400568,
title = {Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging},
author = {Liang, Steven H. and Chen, Jinshan Michael and Normandin, Marc D. and Chang, Jeanne S. and Chang, George C. and Taylor, Christine K. and Trapa, Patrick and Plummer, Mark S. and Para, Kimberly S. and Conn, Edward L. and Lopresti-Morrow, Lori and Lanyon, Lorraine F. and Cook, James M. and Richter, Karl E. G. and Nolan, Charlie E. and Schachter, Joel B. and Janat, Fouad and Che, Ye and Shanmugasundaram, Veerabahu and Lefker, Bruce A. and Enerson, Bradley E. and Livni, Elijahu and Wang, Lu and Guehl, Nicolas J. and Patnaik, Debasis and Wagner, Florence F. and Perlis, Roy and Holson, Edward B. and Haggarty, Stephen J. and El Fakhri, Georges and Kurumbail, Ravi G. and Vasdev, Neil},
abstractNote = {},
doi = {10.1002/anie.201603797},
journal = {Angewandte Chemie (International Edition)},
number = 33,
volume = 55,
place = {Germany},
year = {2016},
month = {6}
}

Journal Article:
Free Publicly Available Full Text
Publisher's Version of Record
DOI: 10.1002/anie.201603797

Citation Metrics:
Cited by: 13 works
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