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Title: Copper-Mediated Radiofluorination of Arylstannanes with [ 18 F]KF

Authors:
 [1];  [2];  [2];  [1];  [3]
  1. Univ. of Michigan, Ann Arbor, MI (United States). Dept. of Chemistry
  2. Univ. of Michigan Medical School, Ann Arbor, MI (United States). Dept. of Radiology
  3. Univ. of Michigan Medical School, Ann Arbor, MI (United States). Dept. of Radiology and the Interdepartmental Program in Medicinal Chemistry
Publication Date:
Research Org.:
Univ. of Michigan Medical School, Ann Arbor, MI (United States)
Sponsoring Org.:
USDOE; National Institutes of Health (NIH); Merck and Company, Inc., Kenilworth, NJ (United States)
OSTI Identifier:
1328258
Alternate Identifier(s):
OSTI ID: 1425388
Grant/Contract Number:  
SC0012484; R01EB021155
Resource Type:
Published Article
Journal Name:
Organic Letters
Additional Journal Information:
Journal Name: Organic Letters Journal Volume: 18 Journal Issue: 20; Journal ID: ISSN 1523-7060
Publisher:
American Chemical Society
Country of Publication:
United States
Language:
English
Subject:
38 RADIATION CHEMISTRY, RADIOCHEMISTRY, AND NUCLEAR CHEMISTRY

Citation Formats

Makaravage, Katarina J., Brooks, Allen F., Mossine, Andrew V., Sanford, Melanie S., and Scott, Peter J. H. Copper-Mediated Radiofluorination of Arylstannanes with [ 18 F]KF. United States: N. p., 2016. Web. doi:10.1021/acs.orglett.6b02911.
Makaravage, Katarina J., Brooks, Allen F., Mossine, Andrew V., Sanford, Melanie S., & Scott, Peter J. H. Copper-Mediated Radiofluorination of Arylstannanes with [ 18 F]KF. United States. doi:10.1021/acs.orglett.6b02911.
Makaravage, Katarina J., Brooks, Allen F., Mossine, Andrew V., Sanford, Melanie S., and Scott, Peter J. H. Mon . "Copper-Mediated Radiofluorination of Arylstannanes with [ 18 F]KF". United States. doi:10.1021/acs.orglett.6b02911.
@article{osti_1328258,
title = {Copper-Mediated Radiofluorination of Arylstannanes with [ 18 F]KF},
author = {Makaravage, Katarina J. and Brooks, Allen F. and Mossine, Andrew V. and Sanford, Melanie S. and Scott, Peter J. H.},
abstractNote = {},
doi = {10.1021/acs.orglett.6b02911},
journal = {Organic Letters},
number = 20,
volume = 18,
place = {United States},
year = {2016},
month = {10}
}

Journal Article:
Free Publicly Available Full Text
Publisher's Version of Record
DOI: 10.1021/acs.orglett.6b02911

Citation Metrics:
Cited by: 16 works
Citation information provided by
Web of Science

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Works referencing / citing this record:

Carbon-Fluorine Reductive Elimination from Nickel(III) Complexes
journal, May 2017

  • Lee, Heejun; Börgel, Jonas; Ritter, Tobias
  • Angewandte Chemie International Edition, Vol. 56, Issue 24
  • DOI: 10.1002/anie.201701552

[Rh III (Cp*)]-catalyzed arylfluorination of α-diazoketoesters for facile synthesis of α-aryl-α-fluoroketoesters
journal, January 2019

  • Ng, Fo-Ning; Chan, Chun-Ming; Li, Jianbin
  • Organic & Biomolecular Chemistry, Vol. 17, Issue 5
  • DOI: 10.1039/c8ob02801j

Baeyer-Villiger oxidation tuned to chemoselective conversion of non-activated [ 18 F]fluorobenzaldehydes to [ 18 F]fluorophenols
journal, June 2019

  • Ermert, Johannes; Castillo Meleán, Johnny; Humpert, Swen
  • Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 62, Issue 8
  • DOI: 10.1002/jlcr.3740

Fast and efficient copper-mediated 18F-fluorination of arylstannanes, aryl boronic acids, and aryl boronic esters without azeotropic drying
journal, October 2019

  • Lahdenpohja, Salla Orvokki; Rajala, Noora Annika; Rajander, Johan
  • EJNMMI Radiopharmacy and Chemistry, Vol. 4, Issue 1
  • DOI: 10.1186/s41181-019-0079-y

Carbon-Fluorine Reductive Elimination from Nickel(III) Complexes
journal, May 2017

  • Lee, Heejun; Börgel, Jonas; Ritter, Tobias
  • Angewandte Chemie International Edition, Vol. 56, Issue 24
  • DOI: 10.1002/anie.201701552

Automated synthesis of PET radiotracers by copper-mediated 18 F-fluorination of organoborons: Importance of the order of addition and competing protodeborylation
journal, February 2018

  • Mossine, Andrew V.; Brooks, Allen F.; Bernard-Gauthier, Vadim
  • Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 61, Issue 3
  • DOI: 10.1002/jlcr.3583

Baeyer-Villiger oxidation tuned to chemoselective conversion of non-activated [ 18 F]fluorobenzaldehydes to [ 18 F]fluorophenols
journal, June 2019

  • Ermert, Johannes; Castillo Meleán, Johnny; Humpert, Swen
  • Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 62, Issue 8
  • DOI: 10.1002/jlcr.3740

[Rh III (Cp*)]-catalyzed arylfluorination of α-diazoketoesters for facile synthesis of α-aryl-α-fluoroketoesters
journal, January 2019

  • Ng, Fo-Ning; Chan, Chun-Ming; Li, Jianbin
  • Organic & Biomolecular Chemistry, Vol. 17, Issue 5
  • DOI: 10.1039/c8ob02801j

Fast and efficient copper-mediated 18F-fluorination of arylstannanes, aryl boronic acids, and aryl boronic esters without azeotropic drying
journal, October 2019

  • Lahdenpohja, Salla Orvokki; Rajala, Noora Annika; Rajander, Johan
  • EJNMMI Radiopharmacy and Chemistry, Vol. 4, Issue 1
  • DOI: 10.1186/s41181-019-0079-y