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Title: Synthesis of [ 18 F]Arenes via the Copper-Mediated [ 18 F]Fluorination of Boronic Acids

Authors:
 [1];  [1];  [2];  [3];  [2];  [2];  [4]
  1. Department of Radiology, University of Michigan Medical School, 1301 Catherine Street, Ann Arbor, Michigan 48109, United States
  2. Department of Chemistry, University of Michigan, 930 North University Avenue, Ann Arbor, Michigan 48109, United States
  3. Department of Medicinal Chemistry, University of Michigan, 428 Church Street, Ann Arbor, Michigan 48109, United States
  4. Department of Radiology, University of Michigan Medical School, 1301 Catherine Street, Ann Arbor, Michigan 48109, United States, Department of Medicinal Chemistry, University of Michigan, 428 Church Street, Ann Arbor, Michigan 48109, United States
Publication Date:
Research Org.:
Univ. of Michigan, Ann Arbor, MI (United States)
Sponsoring Org.:
USDOE Office of Science (SC)
OSTI Identifier:
1225990
Alternate Identifier(s):
OSTI ID: 1345033
Grant/Contract Number:  
SC0012484
Resource Type:
Published Article
Journal Name:
Organic Letters
Additional Journal Information:
Journal Name: Organic Letters Journal Volume: 17 Journal Issue: 23; Journal ID: ISSN 1523-7060
Publisher:
American Chemical Society
Country of Publication:
United States
Language:
English
Subject:
37 INORGANIC, ORGANIC, PHYSICAL, AND ANALYTICAL CHEMISTRY

Citation Formats

Mossine, Andrew V., Brooks, Allen F., Makaravage, Katarina J., Miller, Jason M., Ichiishi, Naoko, Sanford, Melanie S., and Scott, Peter J. H. Synthesis of [ 18 F]Arenes via the Copper-Mediated [ 18 F]Fluorination of Boronic Acids. United States: N. p., 2015. Web. doi:10.1021/acs.orglett.5b02875.
Mossine, Andrew V., Brooks, Allen F., Makaravage, Katarina J., Miller, Jason M., Ichiishi, Naoko, Sanford, Melanie S., & Scott, Peter J. H. Synthesis of [ 18 F]Arenes via the Copper-Mediated [ 18 F]Fluorination of Boronic Acids. United States. doi:10.1021/acs.orglett.5b02875.
Mossine, Andrew V., Brooks, Allen F., Makaravage, Katarina J., Miller, Jason M., Ichiishi, Naoko, Sanford, Melanie S., and Scott, Peter J. H. Sat . "Synthesis of [ 18 F]Arenes via the Copper-Mediated [ 18 F]Fluorination of Boronic Acids". United States. doi:10.1021/acs.orglett.5b02875.
@article{osti_1225990,
title = {Synthesis of [ 18 F]Arenes via the Copper-Mediated [ 18 F]Fluorination of Boronic Acids},
author = {Mossine, Andrew V. and Brooks, Allen F. and Makaravage, Katarina J. and Miller, Jason M. and Ichiishi, Naoko and Sanford, Melanie S. and Scott, Peter J. H.},
abstractNote = {},
doi = {10.1021/acs.orglett.5b02875},
journal = {Organic Letters},
number = 23,
volume = 17,
place = {United States},
year = {2015},
month = {11}
}

Journal Article:
Free Publicly Available Full Text
Publisher's Version of Record
DOI: 10.1021/acs.orglett.5b02875

Citation Metrics:
Cited by: 36 works
Citation information provided by
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Works referencing / citing this record:

Efficient Pathway for the Preparation of Aryl(isoquinoline)iodonium(III) Salts and Synthesis of Radiofluorinated Isoquinolines
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  • Zlatopolskiy, Boris D.; Zischler, Johannes; Krapf, Philipp
  • Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 62, Issue 8
  • DOI: 10.1002/jlcr.3776

Fast and efficient copper-mediated 18F-fluorination of arylstannanes, aryl boronic acids, and aryl boronic esters without azeotropic drying
journal, October 2019

  • Lahdenpohja, Salla Orvokki; Rajala, Noora Annika; Rajander, Johan
  • EJNMMI Radiopharmacy and Chemistry, Vol. 4, Issue 1
  • DOI: 10.1186/s41181-019-0079-y

Efficient Pathway for the Preparation of Aryl(isoquinoline)iodonium(III) Salts and Synthesis of Radiofluorinated Isoquinolines
journal, August 2016

  • Yuan, Zheliang; Cheng, Ran; Chen, Pinhong
  • Angewandte Chemie International Edition, Vol. 55, Issue 39
  • DOI: 10.1002/anie.201606381

One-step synthesis of 4-[ 18 F]fluorobenzyltriphenylphosphonium cation for imaging with positron emission tomography : One-step synthesis of
journal, August 2016

  • Zhang, Zhengxing; Zhang, Chengcheng; Lau, Joseph
  • Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 59, Issue 11
  • DOI: 10.1002/jlcr.3436

Automated synthesis of PET radiotracers by copper-mediated 18 F-fluorination of organoborons: Importance of the order of addition and competing protodeborylation
journal, February 2018

  • Mossine, Andrew V.; Brooks, Allen F.; Bernard-Gauthier, Vadim
  • Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 61, Issue 3
  • DOI: 10.1002/jlcr.3583

Minimalist approach meets green chemistry: Synthesis of 18 F- labeled (hetero)aromatics in pure ethanol
journal, June 2019

  • Zlatopolskiy, Boris D.; Zischler, Johannes; Krapf, Philipp
  • Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 62, Issue 8
  • DOI: 10.1002/jlcr.3776

Fast and efficient copper-mediated 18F-fluorination of arylstannanes, aryl boronic acids, and aryl boronic esters without azeotropic drying
journal, October 2019

  • Lahdenpohja, Salla Orvokki; Rajala, Noora Annika; Rajander, Johan
  • EJNMMI Radiopharmacy and Chemistry, Vol. 4, Issue 1
  • DOI: 10.1186/s41181-019-0079-y