Abstract
The title compound [{sup 14}C]BAY u 3405 (1) was synthesized as part of 8-step sequence. Starting from [U-{sup 14}C]aniline hydrogensulfate the final product 1 was obtained with a specific activity of 741 MBq/mmol (20 mCi/mmol) and a radiochemical purity of > 98 % in an overall yield of 6 and 10 % depending on the method. (author).
Radtke, M;
Boberg, M;
Pleiss, U;
[1]
Rosentreter, U
[2]
- Inst. of Pharmacokinetics, Bayer AG, Wuppertal (Germany)
- Pharma Production, Bayer AG. Wuppertal (Germany)
Citation Formats
Radtke, M, Boberg, M, Pleiss, U, and Rosentreter, U.
Synthesis of (+)-(3R)-3-(4-fluorophenylsulfonamido)-1,2,3,4-tetrahydro-9-[5,6,7,8,12,13-u-{sup 14}C]carbazoleppropanoic acid, [{sup 14}C]BAY u 3405.
United Kingdom: N. p.,
1994.
Web.
doi:10.1002/jlcr.2580341210.
Radtke, M, Boberg, M, Pleiss, U, & Rosentreter, U.
Synthesis of (+)-(3R)-3-(4-fluorophenylsulfonamido)-1,2,3,4-tetrahydro-9-[5,6,7,8,12,13-u-{sup 14}C]carbazoleppropanoic acid, [{sup 14}C]BAY u 3405.
United Kingdom.
https://doi.org/10.1002/jlcr.2580341210
Radtke, M, Boberg, M, Pleiss, U, and Rosentreter, U.
1994.
"Synthesis of (+)-(3R)-3-(4-fluorophenylsulfonamido)-1,2,3,4-tetrahydro-9-[5,6,7,8,12,13-u-{sup 14}C]carbazoleppropanoic acid, [{sup 14}C]BAY u 3405."
United Kingdom.
https://doi.org/10.1002/jlcr.2580341210.
@misc{etde_30627,
title = {Synthesis of (+)-(3R)-3-(4-fluorophenylsulfonamido)-1,2,3,4-tetrahydro-9-[5,6,7,8,12,13-u-{sup 14}C]carbazoleppropanoic acid, [{sup 14}C]BAY u 3405}
author = {Radtke, M, Boberg, M, Pleiss, U, and Rosentreter, U}
abstractNote = {The title compound [{sup 14}C]BAY u 3405 (1) was synthesized as part of 8-step sequence. Starting from [U-{sup 14}C]aniline hydrogensulfate the final product 1 was obtained with a specific activity of 741 MBq/mmol (20 mCi/mmol) and a radiochemical purity of > 98 % in an overall yield of 6 and 10 % depending on the method. (author).}
doi = {10.1002/jlcr.2580341210}
journal = []
issue = {12}
volume = {34}
journal type = {AC}
place = {United Kingdom}
year = {1994}
month = {Dec}
}
title = {Synthesis of (+)-(3R)-3-(4-fluorophenylsulfonamido)-1,2,3,4-tetrahydro-9-[5,6,7,8,12,13-u-{sup 14}C]carbazoleppropanoic acid, [{sup 14}C]BAY u 3405}
author = {Radtke, M, Boberg, M, Pleiss, U, and Rosentreter, U}
abstractNote = {The title compound [{sup 14}C]BAY u 3405 (1) was synthesized as part of 8-step sequence. Starting from [U-{sup 14}C]aniline hydrogensulfate the final product 1 was obtained with a specific activity of 741 MBq/mmol (20 mCi/mmol) and a radiochemical purity of > 98 % in an overall yield of 6 and 10 % depending on the method. (author).}
doi = {10.1002/jlcr.2580341210}
journal = []
issue = {12}
volume = {34}
journal type = {AC}
place = {United Kingdom}
year = {1994}
month = {Dec}
}