Process for the preparation of protected 3-amino-1,2-dihydroxypropane acetal and derivatives thereof
Abstract
A process for producing protected 3-amino-1,2-dihydroxypropane acetal, particularly in chiral forms, for use as an intermediate in the preparation of various 3-carbon compounds which are chiral. In particular, the present invention relates to the process for preparation of 3-amino-1,2-dihydroxypropane isopropylidene acetal. The protected 3-amino-1,2-dihydroxypropane acetal is a key intermediate to the preparation of chiral 3-carbon compounds which in turn are intermediates to various pharmaceuticals.
- Inventors:
-
- Haslett, MI
- East Lansing, MI
- Issue Date:
- Research Org.:
- Michigan State Univ., East Lansing, MI (United States)
- OSTI Identifier:
- 872924
- Patent Number(s):
- 6040464
- Assignee:
- Board of Trustees operating Michigan State University (East Lansing, MI)
- Patent Classifications (CPCs):
-
C - CHEMISTRY C07 - ORGANIC CHEMISTRY C07B - GENERAL METHODS OF ORGANIC CHEMISTRY
C - CHEMISTRY C07 - ORGANIC CHEMISTRY C07C - ACYCLIC OR CARBOCYCLIC COMPOUNDS
- DOE Contract Number:
- FG02-89ER14029
- Resource Type:
- Patent
- Country of Publication:
- United States
- Language:
- English
- Subject:
- process; preparation; protected; 3-amino-1; 2-dihydroxypropane; acetal; derivatives; producing; particularly; chiral; forms; intermediate; various; 3-carbon; compounds; particular; relates; isopropylidene; key; intermediates; pharmaceuticals; carbon compound; chiral form; carbon compounds; /999/
Citation Formats
Hollingsworth, Rawle I, and Wang, Guijun. Process for the preparation of protected 3-amino-1,2-dihydroxypropane acetal and derivatives thereof. United States: N. p., 2000.
Web.
Hollingsworth, Rawle I, & Wang, Guijun. Process for the preparation of protected 3-amino-1,2-dihydroxypropane acetal and derivatives thereof. United States.
Hollingsworth, Rawle I, and Wang, Guijun. Sat .
"Process for the preparation of protected 3-amino-1,2-dihydroxypropane acetal and derivatives thereof". United States. https://www.osti.gov/servlets/purl/872924.
@article{osti_872924,
title = {Process for the preparation of protected 3-amino-1,2-dihydroxypropane acetal and derivatives thereof},
author = {Hollingsworth, Rawle I and Wang, Guijun},
abstractNote = {A process for producing protected 3-amino-1,2-dihydroxypropane acetal, particularly in chiral forms, for use as an intermediate in the preparation of various 3-carbon compounds which are chiral. In particular, the present invention relates to the process for preparation of 3-amino-1,2-dihydroxypropane isopropylidene acetal. The protected 3-amino-1,2-dihydroxypropane acetal is a key intermediate to the preparation of chiral 3-carbon compounds which in turn are intermediates to various pharmaceuticals.},
doi = {},
journal = {},
number = ,
volume = ,
place = {United States},
year = {2000},
month = {1}
}
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