Urea/carbamates FAAH MAGL or dual FAAH/MAGL inhibitors and uses thereof
Abstract
Disclosed are compounds that may be used to inhibit the action of fatty acid amide hydrolase (FAAH), monoacylglycerol lipase (MAGL) or dual FAAH/MAGL. More particularly, compounds of formula II ##STR00001## have utility in a variety of therapeutic uses such as treatment of pain, inflammation, neuropathy, or appetite disorder.
- Inventors:
- Issue Date:
- Research Org.:
- Northeastern Univ., Boston, MA (United States)
- Sponsoring Org.:
- USDOE
- OSTI Identifier:
- 1632602
- Patent Number(s):
- 10570146
- Application Number:
- 15/328,428
- Assignee:
- Northeastern University (Boston, MA)
- Patent Classifications (CPCs):
-
C - CHEMISTRY C07 - ORGANIC CHEMISTRY C07D - HETEROCYCLIC COMPOUNDS
- DOE Contract Number:
- FG02-00ER45852
- Resource Type:
- Patent
- Resource Relation:
- Patent File Date: 07/24/2015
- Country of Publication:
- United States
- Language:
- English
- Subject:
- 59 BASIC BIOLOGICAL SCIENCES; 37 INORGANIC, ORGANIC, PHYSICAL, AND ANALYTICAL CHEMISTRY
Citation Formats
Makriyannis, Alexandros, Shukla, Vidyanand G., and Alapafuja, Shakiru O. Urea/carbamates FAAH MAGL or dual FAAH/MAGL inhibitors and uses thereof. United States: N. p., 2020.
Web.
Makriyannis, Alexandros, Shukla, Vidyanand G., & Alapafuja, Shakiru O. Urea/carbamates FAAH MAGL or dual FAAH/MAGL inhibitors and uses thereof. United States.
Makriyannis, Alexandros, Shukla, Vidyanand G., and Alapafuja, Shakiru O. Tue .
"Urea/carbamates FAAH MAGL or dual FAAH/MAGL inhibitors and uses thereof". United States. https://www.osti.gov/servlets/purl/1632602.
@article{osti_1632602,
title = {Urea/carbamates FAAH MAGL or dual FAAH/MAGL inhibitors and uses thereof},
author = {Makriyannis, Alexandros and Shukla, Vidyanand G. and Alapafuja, Shakiru O.},
abstractNote = {Disclosed are compounds that may be used to inhibit the action of fatty acid amide hydrolase (FAAH), monoacylglycerol lipase (MAGL) or dual FAAH/MAGL. More particularly, compounds of formula II ##STR00001## have utility in a variety of therapeutic uses such as treatment of pain, inflammation, neuropathy, or appetite disorder.},
doi = {},
journal = {},
number = ,
volume = ,
place = {United States},
year = {2020},
month = {2}
}
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