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Title: Tricyclic gyrase inhibitors

Abstract

Disclosed herein are compounds having the structure of Formula I and pharmaceutically suitable salts, esters, and prodrugs thereof that are useful as antibacterially effective tricyclic gyrase inhibitors.Related pharmaceutical compositions, uses and methods of making the compounds are also contemplated.

Inventors:
; ; ; ; ; ; ; ; ; ; ; ; ; ;
Issue Date:
Research Org.:
Lawrence Livermore National Lab. (LLNL), Livermore, CA (United States)
Sponsoring Org.:
USDOE
OSTI Identifier:
1532007
Patent Number(s):
9,732,083
Application Number:
13/496,188
Assignee:
Merck Sharp & Dohme Corp. (New York, NY); Lawrence Livermore National Security, LLC (Livermore, CA)
DOE Contract Number:  
HHSN272200800042C; TC02128.0
Resource Type:
Patent
Resource Relation:
Patent File Date: 2012-03-14
Country of Publication:
United States
Language:
English

Citation Formats

Bensen, Daniel, Chen, Zhiyong, Finn, John, Lam, Thanh To, Lee, Suk Joong, Li, Xiaoming, Phillipson, Douglas W., Tari, Leslie William, Trzoss, Michael, Zhang, Junhu, Lightstone, Felice C., Nguyen, Toan B., Wong, Sergio E., Aristoff, Paul, and Jung, Michael. Tricyclic gyrase inhibitors. United States: N. p., 2017. Web.
Bensen, Daniel, Chen, Zhiyong, Finn, John, Lam, Thanh To, Lee, Suk Joong, Li, Xiaoming, Phillipson, Douglas W., Tari, Leslie William, Trzoss, Michael, Zhang, Junhu, Lightstone, Felice C., Nguyen, Toan B., Wong, Sergio E., Aristoff, Paul, & Jung, Michael. Tricyclic gyrase inhibitors. United States.
Bensen, Daniel, Chen, Zhiyong, Finn, John, Lam, Thanh To, Lee, Suk Joong, Li, Xiaoming, Phillipson, Douglas W., Tari, Leslie William, Trzoss, Michael, Zhang, Junhu, Lightstone, Felice C., Nguyen, Toan B., Wong, Sergio E., Aristoff, Paul, and Jung, Michael. Tue . "Tricyclic gyrase inhibitors". United States. https://www.osti.gov/servlets/purl/1532007.
@article{osti_1532007,
title = {Tricyclic gyrase inhibitors},
author = {Bensen, Daniel and Chen, Zhiyong and Finn, John and Lam, Thanh To and Lee, Suk Joong and Li, Xiaoming and Phillipson, Douglas W. and Tari, Leslie William and Trzoss, Michael and Zhang, Junhu and Lightstone, Felice C. and Nguyen, Toan B. and Wong, Sergio E. and Aristoff, Paul and Jung, Michael},
abstractNote = {Disclosed herein are compounds having the structure of Formula I and pharmaceutically suitable salts, esters, and prodrugs thereof that are useful as antibacterially effective tricyclic gyrase inhibitors.Related pharmaceutical compositions, uses and methods of making the compounds are also contemplated.},
doi = {},
journal = {},
number = ,
volume = ,
place = {United States},
year = {2017},
month = {8}
}

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