Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist

Udompholkul, Parima; Garza-Granados, Ana; Alboreggia, Giulia; Baggio, Carlo; McGuire, Jack; Pegan, Scott D.; Pellecchia, Maurizio

doi:10.1021/acs.jmedchem.3c00467

Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist

Journal Article · 01 June 2023 · Journal of Medicinal Chemistry

DOI:https://doi.org/10.1021/acs.jmedchem.3c00467· OSTI ID:2423308

Udompholkul, Parima ^[1]; Garza-Granados, Ana ^[1]; Alboreggia, Giulia ^[1]; Baggio, Carlo ^[1]; McGuire, Jack ^[1]; Pegan, Scott D. ^[1]; ^[1]

Division of Biomedical Sciences, School of Medicine, University of California, Riverside, 900 University Avenue, Riverside, California 92521, United States

Not provided.

Research Organization:: Argonne National Laboratory (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Organization:: USDOE

DOE Contract Number:: AC02-06CH11357

OSTI ID:: 2423308

Journal Information:: Journal of Medicinal Chemistry, Journal Name: Journal of Medicinal Chemistry Journal Issue: 12 Vol. 66; ISSN 0022-2623

Publisher:: American Chemical Society (ACS)

Country of Publication:: United States

Language:: English

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