Phenylsulfamoyl Benzoic Acid Inhibitor of ERAP2 with a Novel Mode of Inhibition

Arya, Richa; Maben, Zachary; Rane, Digamber; Ali, Akbar; Stern, Lawrence J.

doi:10.1021/acschembio.2c00093

Phenylsulfamoyl Benzoic Acid Inhibitor of ERAP2 with a Novel Mode of Inhibition

Journal Article · 29 June 2022 · ACS Chemical Biology

DOI:https://doi.org/10.1021/acschembio.2c00093· OSTI ID:1982016

Arya, Richa ^[1]; Maben, Zachary ^[1]; Rane, Digamber ^[2]; ^[3]; ^[4]

Department of Pathology, University of Massachusetts Chan Medical School, Worcester, Massachusetts 01655, United States
Kansas University Specialized Chemistry Center, Lawrence, Kansas 66047, United States
Department of Biochemistry & Molecular Pharmacology, University of Massachusetts Chan Medical School, Worcester, Massachusetts 01655, United States
Department of Pathology, University of Massachusetts Chan Medical School, Worcester, Massachusetts 01655, United States; Department of Biochemistry & Molecular Pharmacology, University of Massachusetts Chan Medical School, Worcester, Massachusetts 01655, United States

Not provided.

Research Organization:: Brookhaven National Lab. (BNL), Upton, NY (United States). National Synchrotron Light Source II (NSLS-II)

Sponsoring Organization:: USDOE Office of Science (SC)

DOE Contract Number:: SC0012704

OSTI ID:: 1982016

Journal Information:: ACS Chemical Biology, Vol. 17, Issue 7; ISSN 1554-8929

Publisher:: American Chemical Society (ACS)

Country of Publication:: United States

Language:: English

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