Venglustat Inhibits Protein N-Terminal Methyltransferase 1 in a Substrate-Competitive Manner

Dong, Guangping; Deng, Youchao; Yasgar, Adam; Yadav, Ravi; Talley, Daniel; Zakharov, Alexey V.; Jain, Sankalp; Rai, Ganesha; Noinaj, Nicholas; Simeonov, Anton; Huang, Rong

doi:10.1021/acs.jmedchem.2c01050

Venglustat Inhibits Protein N-Terminal Methyltransferase 1 in a Substrate-Competitive Manner

Journal Article · 01 September 2022 · J. Med. Chem.

DOI:https://doi.org/10.1021/acs.jmedchem.2c01050· OSTI ID:1901249

Dong, Guangping; Deng, Youchao; Yasgar, Adam; Yadav, Ravi; Talley, Daniel; Zakharov, Alexey V.; Jain, Sankalp; Rai, Ganesha; Noinaj, Nicholas; Simeonov, Anton; Huang, Rong

Research Organization:: Advanced Photon Source (APS), Argonne National Laboratory (ANL), Argonne, IL (US)

Sponsoring Organization:: DOE - Office Of Science; NIH; UNIVERSITY

OSTI ID:: 1901249

Journal Information:: J. Med. Chem., Journal Name: J. Med. Chem. Journal Issue: (18) Vol. 65

Country of Publication:: United States

Language:: ENGLISH

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