Discovery and Structural Characterization of Small Molecule Binders of the Human CTLH E3 Ligase Subu

Chana, Chetan K.; Maisonneuve, Pierre; Posternak, Ganna; Grinberg, Nicolas G.A.; Poirson, Juline; Ona, Samara M.; Ceccarelli, Derek F.; Mader, Pavel; St-Cyr, Daniel J.; Pau, Victor; Kurinov, Igor; Tang, Xiaojing; Deng, Dongjing; Cui, Weiren; Su, Wenji; Kuai, Letian; Soll, Richard; Tyers, Mike; Rost, Hannes L.; Batey, Robert A.; Taipale, Mikko; Gingras, Anne-Claude; Sicheri, Frank

doi:10.1021/acs.jmedchem.2c00509

Title: Discovery and Structural Characterization of Small Molecule Binders of the Human CTLH E3 Ligase Subu

Journal Article · 01 September 2022 · J. Med. Chem.

DOI:https://doi.org/10.1021/acs.jmedchem.2c00509· OSTI ID:1901190

Chana, Chetan K.; Maisonneuve, Pierre; Posternak, Ganna; Grinberg, Nicolas G.A.; Poirson, Juline; Ona, Samara M.; Ceccarelli, Derek F.; Mader, Pavel; St-Cyr, Daniel J.; Pau, Victor; Kurinov, Igor; Tang, Xiaojing; Deng, Dongjing; Cui, Weiren; Su, Wenji; Kuai, Letian; Soll, Richard; Tyers, Mike; Rost, Hannes L.; Batey, Robert A. more »

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Research Organization:: Argonne National Laboratory (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Organization:: DOE - Office Of Science; FOREIGN

OSTI ID:: 1901190

Journal Information:: J. Med. Chem., Vol. 65, Issue (19)

Country of Publication:: United States

Language:: ENGLISH

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