Discovery of potent BET bromodomain 1 stereoselective inhibitors using DNA-encoded chemical library

Modukuri, Ram K.; Yu, Zhifeng; Tan, Zhi; Ta, Hai Minh; Ucisik, Melek Nihan; Jin, Zhuang; Anglin, Justin L.; Sharma, Kiran L.; Nyshadham, Pranavanand; Li, Feng; Riehle, Kevin; Faver, John C.; Duong, Kevin; Nagarajan, Sureshbabu; Simmons, Nicholas; Palmer, Stephen S.; Teng, Mingxing; Young, Damian W.; Yi, Joanna S.; Kim, Choel; Matzuk, Martin M.

doi:10.1073/pnas.2122506119

Discovery of potent BET bromodomain 1 stereoselective inhibitors using DNA-encoded chemical library

Journal Article · 01 January 2022 · Proc. Natl. Acad. Sci. USA

DOI:https://doi.org/10.1073/pnas.2122506119· OSTI ID:1870897

Modukuri, Ram K.; Yu, Zhifeng; Tan, Zhi; Ta, Hai Minh; Ucisik, Melek Nihan; Jin, Zhuang; Anglin, Justin L.; Sharma, Kiran L.; Nyshadham, Pranavanand; Li, Feng; Riehle, Kevin; Faver, John C.; Duong, Kevin; Nagarajan, Sureshbabu; Simmons, Nicholas; Palmer, Stephen S.; Teng, Mingxing; Young, Damian W.; Yi, Joanna S.; Kim, Choel more »

Research Organization:: Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Organization:: DOE - Office Of Science; OTHER

OSTI ID:: 1870897

Journal Information:: Proc. Natl. Acad. Sci. USA, Vol. 119, Issue (22)

Country of Publication:: United States

Language:: ENGLISH

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