Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor

Serafim, Ricardo A.M.; da Silva Santiago, Andre; Schwalm, Martin P.; Hu, Zexi; dos Reis, Caio V.; Takarada, Jessica E.; Mezzomo, Priscila; Massirer, Katlin B.; Kudolo, Mark; Gerstenecker, Stefan; Chaikuad, Apirat; Zender, Lars; Knapp, Stefan; Laufer, Stefan; Cou?ago, Rafael M.; Gehringer, Matthias

doi:10.1021/acs.jmedchem.1c01165

Title: Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor

Journal Article · 01 February 2022 · J. Med. Chem.

DOI:https://doi.org/10.1021/acs.jmedchem.1c01165· OSTI ID:1847130

Serafim, Ricardo A.M.; da Silva Santiago, Andre; Schwalm, Martin P.; Hu, Zexi; dos Reis, Caio V.; Takarada, Jessica E.; Mezzomo, Priscila; Massirer, Katlin B.; Kudolo, Mark; Gerstenecker, Stefan; Chaikuad, Apirat; Zender, Lars; Knapp, Stefan; Laufer, Stefan; Cou?ago, Rafael M.; Gehringer, Matthias

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Research Organization:: Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Organization:: DOE - Office Of Science; National Institutes of Health (NIH)

OSTI ID:: 1847130

Journal Information:: J. Med. Chem., Vol. 65, Issue (4)

Country of Publication:: United States

Language:: ENGLISH

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