Rational Alteration of Pharmacokinetics of Chiral Fluorinated and Deuterated Derivatives of Emixustat for Retinal Therapy

Blum, E; Zhang, J.; Zaluski, J.; Einstein, D.; Korshin, E.; Kubas, A.; Gruzman, A.; Tochtrop, G.; Kiser, P.; Palczewski, K.

doi:10.1021/acs.jmedchem.1c00279

Rational Alteration of Pharmacokinetics of Chiral Fluorinated and Deuterated Derivatives of Emixustat for Retinal Therapy

Journal Article · 01 January 2022 · Journal of Medicinal Chemistry

DOI:https://doi.org/10.1021/acs.jmedchem.1c00279· OSTI ID:1817347

Blum, E; Zhang, J.; Zaluski, J.; Einstein, D.; Korshin, E.; Kubas, A.; Gruzman, A.; Tochtrop, G.; Kiser, P.; Palczewski, K.

Research Organization:: Brookhaven National Laboratory (BNL), Upton, NY (United States)

Sponsoring Organization:: ~OTHER

DOE Contract Number:: SC0012704;

OSTI ID:: 1817347

Report Number(s):: BNL-222059-2021-JACI

Journal Information:: Journal of Medicinal Chemistry, Journal Name: Journal of Medicinal Chemistry Journal Issue: 12 Vol. 64; ISSN 0022-2623

Country of Publication:: United States

Language:: English

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