Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 Inhibitors

Vögerl, K; Ong, N.; Senger, J.; Herp, D.; Schmidtkunz, K.; Marek, M.; Müller, M.; Bartel, K.; Shaik, T.; Porter, N.; Robaa, D.; Christianson, D.; Romier, C.; Sippl, W.; Jung, M.; Bracher, F.

doi:10.1021/acs.jmedchem.8b01090

Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 Inhibitors

Journal Article · 01 January 2022 · Journal of Medicinal Chemistry

DOI:https://doi.org/10.1021/acs.jmedchem.8b01090· OSTI ID:1783955

Vögerl, K; Ong, N.; Senger, J.; Herp, D.; Schmidtkunz, K.; Marek, M.; Müller, M.; Bartel, K.; Shaik, T.; Porter, N.; Robaa, D.; Christianson, D.; Romier, C.; Sippl, W.; Jung, M.; Bracher, F.

Research Organization:: Brookhaven National Lab. (BNL), Upton, NY (United States)

Sponsoring Organization:: ~OTHER

DOE Contract Number:: SC0012704

OSTI ID:: 1783955

Report Number(s):: BNL-221486-2021-JACI

Journal Information:: Journal of Medicinal Chemistry, Vol. 62, Issue 3

Country of Publication:: United States

Language:: English

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