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Title: Structures of Hsp90α and Hsp90β bound to a purine-scaffold inhibitor reveal an exploitable residue for drug selectivity

Authors:
 [1];  [2];  [3];  [3];  [3]; ORCiD logo [1]
  1. Hauptman‐Woodward Medical Research Institute Buffalo New York; Department of Structural BiologyJacobs School of Medicine &, Biomedical Sciences, University at Buffalo Buffalo New York
  2. Hauptman‐Woodward Medical Research Institute Buffalo New York
  3. Program in Chemical Biology and Department of MedicineMemorial Sloan Kettering Cancer Center New York New York
Publication Date:
Research Org.:
Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
Sponsoring Org.:
National Institutes of Health (NIH)
OSTI Identifier:
1577176
Resource Type:
Journal Article
Journal Name:
Proteins
Additional Journal Information:
Journal Volume: 87; Journal Issue: 10; Journal ID: ISSN 0887-3585
Publisher:
Wiley
Country of Publication:
United States
Language:
ENGLISH

Citation Formats

Huck, John D., Que, Nanette L. S., Sharma, Sahil, Taldone, Tony, Chiosis, Gabriela, and Gewirth, Daniel T. Structures of Hsp90α and Hsp90β bound to a purine-scaffold inhibitor reveal an exploitable residue for drug selectivity. United States: N. p., 2019. Web. doi:10.1002/prot.25750.
Huck, John D., Que, Nanette L. S., Sharma, Sahil, Taldone, Tony, Chiosis, Gabriela, & Gewirth, Daniel T. Structures of Hsp90α and Hsp90β bound to a purine-scaffold inhibitor reveal an exploitable residue for drug selectivity. United States. doi:10.1002/prot.25750.
Huck, John D., Que, Nanette L. S., Sharma, Sahil, Taldone, Tony, Chiosis, Gabriela, and Gewirth, Daniel T. Wed . "Structures of Hsp90α and Hsp90β bound to a purine-scaffold inhibitor reveal an exploitable residue for drug selectivity". United States. doi:10.1002/prot.25750.
@article{osti_1577176,
title = {Structures of Hsp90α and Hsp90β bound to a purine-scaffold inhibitor reveal an exploitable residue for drug selectivity},
author = {Huck, John D. and Que, Nanette L. S. and Sharma, Sahil and Taldone, Tony and Chiosis, Gabriela and Gewirth, Daniel T.},
abstractNote = {},
doi = {10.1002/prot.25750},
journal = {Proteins},
issn = {0887-3585},
number = 10,
volume = 87,
place = {United States},
year = {2019},
month = {6}
}

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