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Title: Discovery of N-(1-Acryloylazetidin-3-yl)-2-(1 H-indol-1-yl)acetamides as Covalent Inhibitors of KRAS G12C

Authors:
ORCiD logo;  [1]; ORCiD logo; ; ; ; ORCiD logo;  [1];  [1]; ;  [1]; ; ; ; ; ; ;  [1]; ;  [1] more »;  [1]; ; ; ; ORCiD logo;  [1]; ORCiD logo « less
  1. Carmot Therapeutics, Inc. 740 Heinz Avenue, Berkeley, California 94710, United States
Publication Date:
Research Org.:
Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
Sponsoring Org.:
INDUSTRY
OSTI Identifier:
1577150
Resource Type:
Journal Article
Journal Name:
ACS Medicinal Chemistry Letters
Additional Journal Information:
Journal Volume: 10; Journal Issue: 9; Journal ID: ISSN 1948-5875
Publisher:
American Chemical Society (ACS)
Country of Publication:
United States
Language:
ENGLISH

Citation Formats

Shin, Youngsook, Jeong, Joon Won, Wurz, Ryan P., Achanta, Pragathi, Arvedson, Tara, Bartberger, Michael D., Campuzano, Iain D. G., Fucini, Ray, Hansen, Stig K., Ingersoll, John, Iwig, Jeffrey S., Lipford, J. Russell, Ma, Vu, Kopecky, David J., McCarter, John, San Miguel, Tisha, Mohr, Christopher, Sabet, Sudi, Saiki, Anne Y., Sawayama, Andrew, Sethofer, Steven, Tegley, Christopher M., Volak, Laurie P., Yang, Kevin, Lanman, Brian A., Erlanson, Daniel A., and Cee, Victor J. Discovery of N-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as Covalent Inhibitors of KRAS G12C. United States: N. p., 2019. Web. doi:10.1021/acsmedchemlett.9b00258.
Shin, Youngsook, Jeong, Joon Won, Wurz, Ryan P., Achanta, Pragathi, Arvedson, Tara, Bartberger, Michael D., Campuzano, Iain D. G., Fucini, Ray, Hansen, Stig K., Ingersoll, John, Iwig, Jeffrey S., Lipford, J. Russell, Ma, Vu, Kopecky, David J., McCarter, John, San Miguel, Tisha, Mohr, Christopher, Sabet, Sudi, Saiki, Anne Y., Sawayama, Andrew, Sethofer, Steven, Tegley, Christopher M., Volak, Laurie P., Yang, Kevin, Lanman, Brian A., Erlanson, Daniel A., & Cee, Victor J. Discovery of N-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as Covalent Inhibitors of KRAS G12C. United States. doi:10.1021/acsmedchemlett.9b00258.
Shin, Youngsook, Jeong, Joon Won, Wurz, Ryan P., Achanta, Pragathi, Arvedson, Tara, Bartberger, Michael D., Campuzano, Iain D. G., Fucini, Ray, Hansen, Stig K., Ingersoll, John, Iwig, Jeffrey S., Lipford, J. Russell, Ma, Vu, Kopecky, David J., McCarter, John, San Miguel, Tisha, Mohr, Christopher, Sabet, Sudi, Saiki, Anne Y., Sawayama, Andrew, Sethofer, Steven, Tegley, Christopher M., Volak, Laurie P., Yang, Kevin, Lanman, Brian A., Erlanson, Daniel A., and Cee, Victor J. Tue . "Discovery of N-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as Covalent Inhibitors of KRAS G12C". United States. doi:10.1021/acsmedchemlett.9b00258.
@article{osti_1577150,
title = {Discovery of N-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as Covalent Inhibitors of KRAS G12C},
author = {Shin, Youngsook and Jeong, Joon Won and Wurz, Ryan P. and Achanta, Pragathi and Arvedson, Tara and Bartberger, Michael D. and Campuzano, Iain D. G. and Fucini, Ray and Hansen, Stig K. and Ingersoll, John and Iwig, Jeffrey S. and Lipford, J. Russell and Ma, Vu and Kopecky, David J. and McCarter, John and San Miguel, Tisha and Mohr, Christopher and Sabet, Sudi and Saiki, Anne Y. and Sawayama, Andrew and Sethofer, Steven and Tegley, Christopher M. and Volak, Laurie P. and Yang, Kevin and Lanman, Brian A. and Erlanson, Daniel A. and Cee, Victor J.},
abstractNote = {},
doi = {10.1021/acsmedchemlett.9b00258},
journal = {ACS Medicinal Chemistry Letters},
issn = {1948-5875},
number = 9,
volume = 10,
place = {United States},
year = {2019},
month = {8}
}