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Title: Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927

Authors:
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  1. Genentech
Publication Date:
Research Org.:
Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
Sponsoring Org.:
INDUSTRY
OSTI Identifier:
1562699
Resource Type:
Journal Article
Journal Name:
Bioorg. Med. Chem. Lett.
Additional Journal Information:
Journal Volume: 29; Journal Issue: (16) ; 08, 2019
Country of Publication:
United States
Language:
ENGLISH

Citation Formats

Labadie, Sharada S., Li, Jun, Blake, Robert A., Chang, Jae H., Goodacre, Simon, Hartman, Steven J., Liang, Weiling, Kiefer, James R., Kleinheinz, Tracy, Lai, Tommy, Liao, Jiangpeng, Ortwine, Daniel F., Mody, Vidhi, Ray, Nicholas C., Roussel, Fabien, Vinogradova, Maia, Yeap, Siew Kuen, Zhang, Birong, Zheng, Xiaoping, Zbieg, Jason R., Liang, Jun, Wang, Xiaojing, and WuXi App Tec). Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927. United States: N. p., 2019. Web. doi:10.1016/j.bmcl.2019.07.013.
Labadie, Sharada S., Li, Jun, Blake, Robert A., Chang, Jae H., Goodacre, Simon, Hartman, Steven J., Liang, Weiling, Kiefer, James R., Kleinheinz, Tracy, Lai, Tommy, Liao, Jiangpeng, Ortwine, Daniel F., Mody, Vidhi, Ray, Nicholas C., Roussel, Fabien, Vinogradova, Maia, Yeap, Siew Kuen, Zhang, Birong, Zheng, Xiaoping, Zbieg, Jason R., Liang, Jun, Wang, Xiaojing, & WuXi App Tec). Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927. United States. doi:10.1016/j.bmcl.2019.07.013.
Labadie, Sharada S., Li, Jun, Blake, Robert A., Chang, Jae H., Goodacre, Simon, Hartman, Steven J., Liang, Weiling, Kiefer, James R., Kleinheinz, Tracy, Lai, Tommy, Liao, Jiangpeng, Ortwine, Daniel F., Mody, Vidhi, Ray, Nicholas C., Roussel, Fabien, Vinogradova, Maia, Yeap, Siew Kuen, Zhang, Birong, Zheng, Xiaoping, Zbieg, Jason R., Liang, Jun, Wang, Xiaojing, and WuXi App Tec). Thu . "Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927". United States. doi:10.1016/j.bmcl.2019.07.013.
@article{osti_1562699,
title = {Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927},
author = {Labadie, Sharada S. and Li, Jun and Blake, Robert A. and Chang, Jae H. and Goodacre, Simon and Hartman, Steven J. and Liang, Weiling and Kiefer, James R. and Kleinheinz, Tracy and Lai, Tommy and Liao, Jiangpeng and Ortwine, Daniel F. and Mody, Vidhi and Ray, Nicholas C. and Roussel, Fabien and Vinogradova, Maia and Yeap, Siew Kuen and Zhang, Birong and Zheng, Xiaoping and Zbieg, Jason R. and Liang, Jun and Wang, Xiaojing and WuXi App Tec)},
abstractNote = {},
doi = {10.1016/j.bmcl.2019.07.013},
journal = {Bioorg. Med. Chem. Lett.},
number = (16) ; 08, 2019,
volume = 29,
place = {United States},
year = {2019},
month = {9}
}