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Title: Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A

Authors:
 [1];  [2];  [2];  [3];  [2];  [3]; ORCiD logo [4];  [4];  [4];  [4];  [4];  [4];  [4];  [4];  [4];  [4];  [4];  [4]; ORCiD logo [4];  [4] more »; ; ; ORCiD logo [1] « less
  1. Department of Molecular and Cellular Oncology, The University of Texas MD Anderson Cancer Center, Houston, Texas 77030, United States; Department of Biochemistry, Emory University School of Medicine, Atlanta, Georgia 30322, United States
  2. Department of Molecular and Cellular Oncology, The University of Texas MD Anderson Cancer Center, Houston, Texas 77030, United States
  3. Department of Biochemistry, Emory University School of Medicine, Atlanta, Georgia 30322, United States
  4. National Center for Advancing Translational Sciences, National Institutes of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States
Publication Date:
Research Org.:
Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
Sponsoring Org.:
NCINIH
OSTI Identifier:
1506493
Resource Type:
Journal Article
Journal Name:
Journal of Medicinal Chemistry
Additional Journal Information:
Journal Volume: 61; Journal Issue: 23; Journal ID: ISSN 0022-2623
Publisher:
American Chemical Society (ACS)
Country of Publication:
United States
Language:
ENGLISH

Citation Formats

Horton, John R., Woodcock, Clayton B., Chen, Qin, Liu, Xu, Zhang, Xing, Shanks, John, Rai, Ganesha, Mott, Bryan T., Jansen, Daniel J., Kales, Stephen C., Henderson, Mark J., Cyr, Matthew, Pohida, Katherine, Hu, Xin, Shah, Pranav, Xu, Xin, Jadhav, Ajit, Maloney, David J., Hall, Matthew D., Simeonov, Anton, Fu, Haian, Vertino, Paula M., and Cheng, Xiaodong. Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A. United States: N. p., 2018. Web. doi:10.1021/acs.jmedchem.8b01219.
Horton, John R., Woodcock, Clayton B., Chen, Qin, Liu, Xu, Zhang, Xing, Shanks, John, Rai, Ganesha, Mott, Bryan T., Jansen, Daniel J., Kales, Stephen C., Henderson, Mark J., Cyr, Matthew, Pohida, Katherine, Hu, Xin, Shah, Pranav, Xu, Xin, Jadhav, Ajit, Maloney, David J., Hall, Matthew D., Simeonov, Anton, Fu, Haian, Vertino, Paula M., & Cheng, Xiaodong. Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A. United States. doi:10.1021/acs.jmedchem.8b01219.
Horton, John R., Woodcock, Clayton B., Chen, Qin, Liu, Xu, Zhang, Xing, Shanks, John, Rai, Ganesha, Mott, Bryan T., Jansen, Daniel J., Kales, Stephen C., Henderson, Mark J., Cyr, Matthew, Pohida, Katherine, Hu, Xin, Shah, Pranav, Xu, Xin, Jadhav, Ajit, Maloney, David J., Hall, Matthew D., Simeonov, Anton, Fu, Haian, Vertino, Paula M., and Cheng, Xiaodong. Sat . "Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A". United States. doi:10.1021/acs.jmedchem.8b01219.
@article{osti_1506493,
title = {Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A},
author = {Horton, John R. and Woodcock, Clayton B. and Chen, Qin and Liu, Xu and Zhang, Xing and Shanks, John and Rai, Ganesha and Mott, Bryan T. and Jansen, Daniel J. and Kales, Stephen C. and Henderson, Mark J. and Cyr, Matthew and Pohida, Katherine and Hu, Xin and Shah, Pranav and Xu, Xin and Jadhav, Ajit and Maloney, David J. and Hall, Matthew D. and Simeonov, Anton and Fu, Haian and Vertino, Paula M. and Cheng, Xiaodong},
abstractNote = {},
doi = {10.1021/acs.jmedchem.8b01219},
journal = {Journal of Medicinal Chemistry},
issn = {0022-2623},
number = 23,
volume = 61,
place = {United States},
year = {2018},
month = {11}
}