Structural insights into binding specificity, efficacy and bias of a β2AR partial agonist

Masureel, Matthieu; Zou, Yaozhong; Picard, Louis-Philippe; van der Westhuizen, Emma; Mahoney, Jacob P.; Rodrigues, João P.  G.  L.  M.; Mildorf, Thomas J.; Dror, Ron O.; Shaw, David E.; Bouvier, Michel; Pardon, Els; Steyaert, Jan; Sunahara, Roger K.; Weis, William I.; Zhang, Cheng; Kobilka, Brian K.

doi:10.1038/s41589-018-0145-x

Title: Structural insights into binding specificity, efficacy and bias of a β2AR partial agonist

Journal Article · Tue Oct 16 00:00:00 EDT 2018 · Nature Chemical Biology

DOI:https://doi.org/10.1038/s41589-018-0145-x· OSTI ID:1502205

Masureel, Matthieu; Zou, Yaozhong; Picard, Louis-Philippe;

; Mahoney, Jacob P.; Rodrigues, João P. G. L. M.; Mildorf, Thomas J.; Dror, Ron O.; Shaw, David E.;

; Pardon, Els; Steyaert, Jan;

; Weis, William I.;

; Kobilka, Brian K.

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Research Organization:: Argonne National Laboratory (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Organization:: NIHFOREIGN

OSTI ID:: 1502205

Journal Information:: Nature Chemical Biology, Vol. 14, Issue 11; ISSN 1552-4450

Publisher:: Nature Publishing Group

Country of Publication:: United States

Language:: ENGLISH

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