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Title: Crystal structure of N-{N-[N-acetyl-(S)-leuc­yl]-(S)-leuc­yl}norleucinal (ALLN), an inhibitor of proteasome

Authors:
; ; ;  [1]
  1. NCI
Publication Date:
Research Org.:
Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
Sponsoring Org.:
NCI
OSTI Identifier:
1244725
Resource Type:
Journal Article
Journal Name:
Acta Crystallographica. Section E, Crystallographic Communications
Additional Journal Information:
Journal Volume: 71; Journal Issue: 3; Journal ID: ISSN 2056-9890
Country of Publication:
United States
Language:
ENGLISH

Citation Formats

Czerwinski, A., Basava, C., Dauter, M., Dauter, Z., Peptides), and Leidos). Crystal structure of N-{N-[N-acetyl-(S)-leuc­yl]-(S)-leuc­yl}norleucinal (ALLN), an inhibitor of proteasome. United States: N. p., 2016. Web. doi:10.1107/S2056989015002091.
Czerwinski, A., Basava, C., Dauter, M., Dauter, Z., Peptides), & Leidos). Crystal structure of N-{N-[N-acetyl-(S)-leuc­yl]-(S)-leuc­yl}norleucinal (ALLN), an inhibitor of proteasome. United States. doi:10.1107/S2056989015002091.
Czerwinski, A., Basava, C., Dauter, M., Dauter, Z., Peptides), and Leidos). Fri . "Crystal structure of N-{N-[N-acetyl-(S)-leuc­yl]-(S)-leuc­yl}norleucinal (ALLN), an inhibitor of proteasome". United States. doi:10.1107/S2056989015002091.
@article{osti_1244725,
title = {Crystal structure of N-{N-[N-acetyl-(S)-leuc­yl]-(S)-leuc­yl}norleucinal (ALLN), an inhibitor of proteasome},
author = {Czerwinski, A. and Basava, C. and Dauter, M. and Dauter, Z. and Peptides) and Leidos)},
abstractNote = {},
doi = {10.1107/S2056989015002091},
journal = {Acta Crystallographica. Section E, Crystallographic Communications},
issn = {2056-9890},
number = 3,
volume = 71,
place = {United States},
year = {2016},
month = {7}
}

Works referenced in this record:

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Inhibition of the Ubiquitin-Proteasome System by Natural Products for Cancer Therapy
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Development of proteasome inhibitors as research tools and cancer drugs
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Multiparametric scaling of diffraction intensities
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    Works referencing / citing this record:

    CCDC 1046561: Experimental Crystal Structure Determination: QUBVOA : N-Acetylleucyl-N-(1-oxohexan-2-yl)leucinamide
    dataset, January 2015

    • Czerwinski, A.; Basava, C.; Dauter, M.
    • Cambridge Structural Database (CSD)
    • DOI: 10.5517/cc14411c

    Dysfunction of the ubiquitin-proteasome system in multiple disease conditions: therapeutic approaches
    journal, November 2008


    Covalent complexes of proteasome model with peptide aldehyde inhibitors MG132 and MG101: docking and molecular dynamics study
    journal, May 2009


    Cyclodextrins as templates for the presentation of protease inhibitors
    journal, August 1996


    Proteasome Inhibitors: An Expanding Army Attacking a Unique Target
    journal, January 2012


    20S Proteasome and Its Inhibitors:  Crystallographic Knowledge for Drug Development
    journal, March 2007

    • Borissenko, Ljudmila; Groll, Michael
    • Chemical Reviews, Vol. 107, Issue 3
    • DOI: 10.1021/cr0502504

    Structure of 20S proteasome from yeast at 2.4Å resolution
    journal, April 1997

    • Groll, Michael; Ditzel, Lars; Löwe, Jan
    • Nature, Vol. 386, Issue 6624
    • DOI: 10.1038/386463a0

    Inhibition of the Ubiquitin-Proteasome System by Natural Products for Cancer Therapy
    journal, February 2010


    Development of proteasome inhibitors as research tools and cancer drugs
    journal, November 2012



    journal, February 2010

    • Pietsch, Markus; Chua, Krystle; Abell, Andrew
    • Current Topics in Medicinal Chemistry, Vol. 10, Issue 3
    • DOI: 10.2174/156802610790725489


    journal, February 2010



    journal, December 2011