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Title: Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives

Authors:
; ; ; ; ; ; ; ; ; ; ; ; ; ; ; ;  [1];  [2]
  1. (Takeda Cali)
  2. (
Publication Date:
Research Org.:
Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)
Sponsoring Org.:
INDUSTRY
OSTI Identifier:
1191735
Resource Type:
Journal Article
Journal Name:
J. Med. Chem.
Additional Journal Information:
Journal Volume: 56; Journal Issue: (16) ; 08, 2013
Country of Publication:
United States
Language:
ENGLISH

Citation Formats

Okaniwa, Masanori, Hirose, Masaaki, Arita, Takeo, Yabuki, Masato, Nakamura, Akito, Takagi, Terufumi, Kawamoto, Tomohiro, Uchiyama, Noriko, Sumita, Akihiko, Tsutsumi, Shunichirou, Tottori, Tsuneaki, Inui, Yoshitaka, Sang, Bi-Ching, Yano, Jason, Aertgeerts, Kathleen, Yoshida, Sei, Ishikawa, Tomoyasu, and Takeda). Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives. United States: N. p., 2013. Web. doi:10.1021/jm400778d.
Okaniwa, Masanori, Hirose, Masaaki, Arita, Takeo, Yabuki, Masato, Nakamura, Akito, Takagi, Terufumi, Kawamoto, Tomohiro, Uchiyama, Noriko, Sumita, Akihiko, Tsutsumi, Shunichirou, Tottori, Tsuneaki, Inui, Yoshitaka, Sang, Bi-Ching, Yano, Jason, Aertgeerts, Kathleen, Yoshida, Sei, Ishikawa, Tomoyasu, & Takeda). Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives. United States. doi:10.1021/jm400778d.
Okaniwa, Masanori, Hirose, Masaaki, Arita, Takeo, Yabuki, Masato, Nakamura, Akito, Takagi, Terufumi, Kawamoto, Tomohiro, Uchiyama, Noriko, Sumita, Akihiko, Tsutsumi, Shunichirou, Tottori, Tsuneaki, Inui, Yoshitaka, Sang, Bi-Ching, Yano, Jason, Aertgeerts, Kathleen, Yoshida, Sei, Ishikawa, Tomoyasu, and Takeda). Thu . "Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives". United States. doi:10.1021/jm400778d.
@article{osti_1191735,
title = {Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives},
author = {Okaniwa, Masanori and Hirose, Masaaki and Arita, Takeo and Yabuki, Masato and Nakamura, Akito and Takagi, Terufumi and Kawamoto, Tomohiro and Uchiyama, Noriko and Sumita, Akihiko and Tsutsumi, Shunichirou and Tottori, Tsuneaki and Inui, Yoshitaka and Sang, Bi-Ching and Yano, Jason and Aertgeerts, Kathleen and Yoshida, Sei and Ishikawa, Tomoyasu and Takeda)},
abstractNote = {},
doi = {10.1021/jm400778d},
journal = {J. Med. Chem.},
number = (16) ; 08, 2013,
volume = 56,
place = {United States},
year = {2013},
month = {8}
}