Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor

Biggadike, Keith; Bledsoe, Randy K.; Coe, Diane M.; Cooper, Tony W.J.; House, David; Macdonald, Simon J.F.; Madauss, Kevin P.; McLay, Iain M.; Shipley, Tracy J.; Taylor, Simon J.; Tran, Thuy B.; Uings, Iain J.; Weller, Victoria; Williams, Shawn P.

doi:10.1073/pnas.0909125106

Title: Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor

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Authors:

Biggadike, Keith; Bledsoe, Randy K.; Coe, Diane M.; Cooper, Tony W.J.; House, David; Macdonald, Simon J.F.; Madauss, Kevin P.; McLay, Iain M.; Shipley, Tracy J.; Taylor, Simon J.; Tran, Thuy B.; Uings, Iain J.; Weller, Victoria; Williams, Shawn P. ^[1]

GSKNC

Publication Date:: Wed Aug 13 00:00:00 EDT 2014

Research Org.:: Argonne National Lab. (ANL), Argonne, IL (United States). Advanced Photon Source (APS)

Sponsoring Org.:: INDUSTRY

OSTI Identifier:: 1149625

Resource Type:: Journal Article

Journal Name:: Proc. Natl. Acad. Sci. USA

Additional Journal Information:: Journal Volume: 106; Journal Issue: (43) ; 10, 2009

Country of Publication:: United States

Language:: ENGLISH

Citation Formats


                    Biggadike, Keith, Bledsoe, Randy K., Coe, Diane M., Cooper, Tony W.J., House, David, Iannone, Marie A., Macdonald, Simon J.F., Madauss, Kevin P., McLay, Iain M., Shipley, Tracy J., Taylor, Simon J., Tran, Thuy B., Uings, Iain J., Weller, Victoria, Williams, Shawn P., and GSK). Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor.  United States: N. p., 2014. 
        Web.  doi:10.1073/pnas.0909125106.

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                    Biggadike, Keith, Bledsoe, Randy K., Coe, Diane M., Cooper, Tony W.J., House, David, Iannone, Marie A., Macdonald, Simon J.F., Madauss, Kevin P., McLay, Iain M., Shipley, Tracy J., Taylor, Simon J., Tran, Thuy B., Uings, Iain J., Weller, Victoria, Williams, Shawn P., & GSK). Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor.  United States.  https://doi.org/10.1073/pnas.0909125106

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                    Biggadike, Keith, Bledsoe, Randy K., Coe, Diane M., Cooper, Tony W.J., House, David, Iannone, Marie A., Macdonald, Simon J.F., Madauss, Kevin P., McLay, Iain M., Shipley, Tracy J., Taylor, Simon J., Tran, Thuy B., Uings, Iain J., Weller, Victoria, Williams, Shawn P., and GSK). 2014.  
        "Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor".  United States.  https://doi.org/10.1073/pnas.0909125106.

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@article{osti_1149625,

  title        = {Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor},

  author       = {Biggadike, Keith and Bledsoe, Randy K. and Coe, Diane M. and Cooper, Tony W.J. and House, David and Iannone, Marie A. and Macdonald, Simon J.F. and Madauss, Kevin P. and McLay, Iain M. and Shipley, Tracy J. and Taylor, Simon J. and Tran, Thuy B. and Uings, Iain J. and Weller, Victoria and Williams, Shawn P. and GSK)},

  abstractNote = {},

  doi          = {10.1073/pnas.0909125106},

  url          = {https://www.osti.gov/biblio/1149625},
  journal      = {Proc. Natl. Acad. Sci. USA},
number       = (43) ; 10, 2009,

  volume       = 106,

  place        = {United States},

  year         = {Wed Aug 13 00:00:00 EDT 2014},

  month        = {Wed Aug 13 00:00:00 EDT 2014}

}

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https://doi.org/10.1073/pnas.0909125106

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Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor

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