| Sample search results for: a1 receptor activation |
| 1 | List of Abbreviations Acknowledgments | ||
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Summary: short heterodimer partner SXR steroid X receptor SULT2A1 sulfotransferase 2A1 UW university of wisconsin... export pump BUD budesonide C colon CA cholic acid CAR constitutive active/androstane receptor CDCA... transporter PAR pregnane ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 2 | Bradfield; Mechanisms of Liver Carcinogenesis 18 UNIT VI: Nuclear Receptors: Zn Finger proteins and their roles in | ||
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Summary: homology. Many of these orphans probably not receptors at all, many appear to be constituitively active... activated receptor (PPAR) and vitamin D receptor (VDR) are all bound to chromatin as a heterodimer... GR/PR/MR Receptor Signaling KEY 7) ... |
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Source: Bradfield, Christopher A. - McArdle Laboratory for Cancer , University of Wisconsin at Madison |
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Collection: Biology and Medicine |
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| 3 | This article was originally published in the Encyclopedia of Neuroscience published by Elsevier, and the attached copy is provided by Elsevier for the | ||
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Summary: Four different P1 receptor subtypes, A1, A2A, A2B, and A3, have been cloned. All are G... transmembrane domain (see Figure 1(a)). P1 receptors couple principally to adenylate cy- clase. A1 and A3... for both affinity and activity. The most ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 4 | JOURNAL OF RECEPTORS AND SIGNAL TRANSDUCTION Vol. 24, No. 3, pp. 165205, 2004 | ||
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Summary: phosphatase 1 regulates the activity of many receptors, enzymes, ion channels, and transcription factors. D1... or Golf to mediate D1-like receptor activation of adenylate cyclase. In human embryonic kidney (HEK) 293... 1 receptor activation of adenylate cyclase is ... |
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Source: Neve, Kim A. - Department of Behavioral Neuroscience, Oregon Health and Science University |
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Collection: Biology and Medicine |
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| 5 | Copyright C Blackwell Munksgaard 2002 Traffic 2002; 3: 866877 | ||
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Summary: expressing HA-tagged receptors were treated with agonist (C5a 1mM, 30min) or left untreated. Cells were fixed... -9219 Constitutive Activation and Endocytosis of the Complement Factor 5a Receptor: Evidence for Multiple Activated... constitutively ... |
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Source: Bourne, Henry - Department of Cellular and Molecular Pharmacology, University of California at San Francisco |
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Collection: Biology and Medicine |
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| 6 | P2 receptor web: Complexity and fine-tuning Cinzia Volont a,, Susanna Amadio a | ||
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Summary: et al., 1995). Homomeric P2X4 receptors are activated by ATP, but not by ,-methylene ATP (,-me... receptor is not activated by ,-meATP, and is blocked by 8-(3- benzamido-4-methylbenzamido)-naphthalene-1... the level of intracellular calcium ions: whereas activation of P2X ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 7 | Enhancement of the surface expression of G protein-coupled receptors | ||
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Summary: and functional activity of a1D- adrenergic receptors. J. Pharmacol. Exp. Ther. 313, 1623 38 Bush, C.F. et al... -terminus of the a1D-adrenoceptor (a1D-AR) dramatically enhanced expression of receptor ... |
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Source: Hall, Randy A - Department of Pharmacology, Emory University |
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Collection: Biology and Medicine |
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| 8 | D2/D3 Dopamine Receptor Heterodimers Exhibit Unique Functional Properties* | ||
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Summary: for heterodimerization has recently been provided for dopamine D1 and adenosine A1 receptors as well as for dopamine D2... receptor forms hetero-oligomers with the adenosine A1 receptor. As the issue of G protein-coupled ... |
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Source: Vogel, Zvi - Department of Neurobiology, Weizmann Institute of Science |
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Collection: Biology and Medicine |
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| 9 | Ligand accumulation counteracts therapeutic inhibition of receptor systems | ||
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Summary: - ceptor activation the growth factor molecule is cleared from the environment by receptor mediated... of receptor activation by inhibitory drugs, and its interplay with the ligand con- centration... activation. This is the case for a variety of receptor families ... |
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Source: Duffy, Ken - Hamilton Institute, National University of Ireland, Maynooth |
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Collection: Computer Technologies and Information Sciences |
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| 10 | No evidence for cross-talk between the adenosine A1 and the serotonin-1A receptor system after chronic A1 receptor | ||
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Summary: a decrease in adenosine A1 receptor numbers and an increase in the amount of adenosine A1 receptor-activated... . Particularly, it is known that adenosine A1 and serotonin-1A receptors ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 11 | Heterodimerization of G Protein-Coupled Receptors: Specificity and Functional Significance | ||
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Summary: GPCRs (A1, A2A, A2b, and A3), whereas ATP activates P2X receptors, which are ion channels, as well... heterodimerization between purinergic receptor subtypes has been reported for A1R and P2Y1R in both transfected cells... dopamine ... |
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Source: Hall, Randy A - Department of Pharmacology, Emory University |
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Collection: Biology and Medicine |
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| 12 | J Neural Transm (2007) 114: 4975 DOI 10.1007/s00702-006-0589-0 | ||
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Summary: receptor (see Marshall, 2005). Also the A1R= P2Y1R heteromerization leads to the appearance of an A1... accumbens (Diaz-Cabiale et al., 2001). In higher doses CGS 21680 but not an A1 receptor agonist could antag... ... |
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Source: Chin-Sang, Ian - Department of Biology, Queen's University (Kingston) |
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Collection: Biology and Medicine |
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| 13 | The recently deorphanized GPR80 (GPR99) proposed to be the P2Y15 receptor is not a genuine P2Y receptor | ||
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Summary: the pharmacological characterization of novel receptors. Moreover, adenosine A1 and P2Y1 receptors have been shown... previously to form heterodimers that enable the A1 receptor to bind and respond to ADP [6], and thus... ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 14 | THE TETHERING ARM OF THE EGF RECEPTOR IS REQUIRED FOR NEGATIVE COOPERATIVITY AND SIGNAL TRANSDUCTION | ||
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Summary: exhibited relatively weak kinase activity as compared to the wild type receptor. For the average of four... receptor mediated essentially wild type levels of activation of both MAP kinase (Figure 6B) and Akt (Figure... the tyrosine kinase activity of the receptor, is ... |
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Source: Pike, Linda J. - Department of Biochemistry and Molecular Biophysics, Washington University in St. Louis |
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Collection: Biology and Medicine |
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| 15 | Dual constrictor and dilator actions of ETB receptors in the rat renal microcirculation: interactions with ETA receptors | ||
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Summary: cells (38). Both receptor types are coupled to Gq proteins, thereby activating several signaling... to constriction of smooth muscle cells. Activation of endothelial ETB receptors by the same signaling pathways... antagonists (7 nmol/min, each). Renal hemodynamic response to activation ... |
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Source: Just, Armin - Physiologisches Institut I, Albert-Ludwigs-Universität Freiburg |
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Collection: Biology and Medicine |
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| 16 | Strain zygocity Gene Name Ahr -/-Aryl-hydrocarbon receptor | ||
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Summary: proto-oncogene 1 Aldh5a1 +/- Aldhehyde dehydrogenase family 5, subfamily A1 Alox15 -/- Arachidonate 15... endothelial hyaluronan receptor 1 Lpl -/- Lipoprotein lipase Map2k3 -/- Mitogen-activated protein... -/- Plasminogen activator, ... |
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Source: Silva, Alcino - Department of Neurobiology, University of California at Los Angeles |
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Collection: Biology and Medicine |
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| 17 | Introduction Chapter 1 1 Introduction | ||
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Summary: , 7-TM GPCRs). The receptors are activated upon binding an endogenous neurotransmitter molecule... to describe the activation of GPCRs by means of a ternary complex formed by a receptor, an agonist, and a G... in this thesis to investigate structure as well as function of a recently discovered ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 18 | Interneuron Diversity series Diversity of inhibitory | ||
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Summary: -positive interneurons innervate somatic GABAA receptors with a large a1:a2 subunit ratio [35]. This clear segregation... than receptors containing the a1 subunit [36]. Indeed, in mice lacking the a1 subunit, miniature IPSCs... ... |
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Source: Kalil, Ronald E. - Neuroscience Training Program & W.M. Keck Laboratory for Biological Imaging, University of Wisconsin at Madison |
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Collection: Biology and Medicine |
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| 19 | Brain Research 869 (2000) 178185 www.elsevier.com/locate/bres | ||
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Summary: activity, and period length and integrity of rhythms during exposure to constant light. The receptor... receptors5A with a Leica TCS NT confocal microscope. FITC labeled normally restrains exploratory activity... peptideprotein conju- phase shifts, roles for both 5-HT and the 5-HT ... |
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Source: Kalil, Ronald E. - Neuroscience Training Program & W.M. Keck Laboratory for Biological Imaging, University of Wisconsin at Madison |
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Collection: Biology and Medicine |
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| 20 | Constitutive Activity of a Chimeric D2/D1 Dopamine Receptor LAURA B. KOZELL and KIM A. NEVE | ||
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Summary: Constitutive Activity of a Chimeric D2/D1 Dopamine Receptor LAURA B. KOZELL and KIM A. NEVE... that multiple D2 receptor cytoplasmic domains acting in concert are neces- sary for receptor activation of Gi... of activating Gs. D2[1 4,7] exhibited several ... |
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Source: Neve, Kim A. - Department of Behavioral Neuroscience, Oregon Health and Science University |
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Collection: Biology and Medicine |
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| 21 | 14 Bushan, M. et al. (2002) Anti-E-selectin is ineffective in the treatment of psoriasis: a randomized trial. Br. J. Dermatol. 146, 824831 | ||
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Summary: : a randomized trial. Br. J. Dermatol. 146, 824831 15 Maly, P. et al. (1996) The a(1,3)fucosyltransferase Fuc... that this nucleotide and other related sugar-nucleotides can exert pharmacological activity and thus receptor(s... in P2Y receptor activity From a ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 22 | www.landesbioscience.com Cell Cycle 1 Cell CyCle features Cell CyCle features | ||
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Summary: of transducing signals into the ligand-expressing cells.1 Since Eph receptor EphA1 was origi- nally cloned... Activation of EphA receptors leads to ERK inhibition (probably though RasGAP) and activa- tion of TSC1... www.landesbioscience.com Cell Cycle 1 Cell CyCle features Cell CyCle ... |
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Source: Chin-Sang, Ian - Department of Biology, Queen's University (Kingston) |
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Collection: Biology and Medicine |
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| 23 | doi:10.1152/ajpgi.00147.2006 291:605-610, 2006. First published May 4, 2006;Am J Physiol Gastrointest Liver Physiol | ||
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Summary: , and adenosine A1 receptors) are capable of mediating sustained contraction via sequential activation of PI 3... receptors. Phospholipase C (PLC)- activity and Rho kinase activity were used as markers of pathways... -stimulated ... |
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Source: Hu, Wen-Hui - Department of Physiology, Virginia Commonwealth University |
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Collection: Biology and Medicine |
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| 24 | New Modes of Action for Endocrine-Disrupting Michelle M. Tabb and Bruce Blumberg | ||
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Summary: the transcriptional activity of nuclear receptors by modulating proteasome-mediated degradation of nuclear receptors... , polychlorinated biphenyl; PPAR , peroxisomal proliferator-activated receptor ; RXR, retinoic acid X receptor; SXR... by androgens, estrogens, and ... |
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Source: Blumberg, Bruce - Department of Developmental and Cell Biology, University of California, Irvine |
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Collection: Biology and Medicine |
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| 25 | Purinoceptors on Neuroglia Alexei Verkhrasky & Oleg A. Krishtal & | ||
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Summary: receptors activate cyclic AMP (cAMP) production via Gs proteins. A1 and A3 receptors also regulate phospholi... in rat-cultured astroglia [71]. Activation of A1 receptors in rat-cultured astrocytes ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 26 | The concept of purinergic neurotransmission was pro-posed in 1972 (REF. 1), after it was shown that adenosine | ||
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Summary: inhibitory modulator through P1(A1 ) receptors, but ATP itself can act presynaptically either to inhibit... , and in a rat model of Parkinson's disease, A1 , dopamine D1 and glutamate mGlu5 receptors have been shown... presynaptic ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 27 | doi:10.1152/ajpgi.90285.2008 295:78-87, 2008. First published May 15, 2008;Am J Physiol Gastrointest Liver Physiol | ||
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Summary: -purified antibodies directed against the COOH terminus of the CB2 receptor: CB22-A (1:250, Alpha Diag- nostics, Alpha... the hypothesis that CB2 receptors are expressed in the enteric nervous system and are activated... these facts together, we conclude that ... |
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Source: Buckley, Nancy E. - Biological Sciences Department, California State Polytechnic University at Pomona |
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Collection: Biology and Medicine |
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| 28 | ORIGINAL PAPER P2X receptors are differentially expressed on vasopressin- | ||
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Summary: a direct input originating from A1 cells located in the caudal ven- trolateral medulla in which synapse... receptor, rather than via a voltage-dependent Ca2? channel. These data imply that activation of different... ZP, Levy A, Lightman SL (1994) Activation of specific ATP ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 29 | Purine and pyrimidine receptors G. Burnstock | ||
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Summary: by ectonucleotidases. Four subtypes have been identified, A1, A2A, A2B and A3 receptors. P2 receptors are activated... different P1 receptor subtypes, A1, A2A, A2B and A3, have been cloned and charac- terised [2225]. All... ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 30 | Purine and pyrimidine receptors G. Burnstock | ||
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Summary: , complementary DNAs (cDNAs) encoding two different P1 receptor subtypes (A1 and A2) were isolated [20], and... , shortly after, the A3 subtype was identified [21]. Four different P1 receptor subtypes, A1, A2A, A2B and A... transmembrane domain. Polymorphisms have been ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 31 | NEUROKININ RELEASE IN THE RAT NUCLEUS OF THE SOLITARY TRACT VIA NMDA AND AMPA RECEPTORS | ||
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Summary: in vitro brainstem slices, immunoreactivity for NK1 receptor (Fig. 2A, A1) and NK3 receptors (Fig. 3D... internalization in neurons of the NST. (A^A1) NK1 receptor immunoreactivity is located on the surface of neurons... ), neurokinin A (0.1 WM, ... |
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Source: Cossart, Rosa - Institut de Neurobiologie de la Méditerranée, Inserm |
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Collection: Biology and Medicine |
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| 32 | Current Pharmaceutical Design, 2009, 15, 000-000 1 1381-6128/09 $55.00+.00 2009 Bentham Science Publishers Ltd. | ||
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Summary: also form heterodimeric com- plexes [64] or with other receptors. For example, adenosine A1 receptors... and adenosine A1 receptors have also been shown to form func- tionally interactive heteromeric complexes. D. ATP... (broken red line) to ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 33 | Glucocorticoid receptor physiology Marjet D. Heitzer & Irene M. Wolf & Edwin R. Sanchez & | ||
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Summary: to assist in receptor translocation through the nuclear pore [9]. A second activation function (AF-2) domain... of transcriptionally activated proinflammatory genes. Finally, while manyFig. 1 General schematic of steroid receptor... is the role these TPR proteins play in the regulation of steroid ... |
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Source: Brand, Paul H. - Department of Physiology and Pharmacology, University of Toledo; Toledo, University of - Center for Diabetes and Endocrine Research (CeDER) |
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Collection: Biology and Medicine |
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| 34 | *MRC Laboratory of Molecular Biology, | ||
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Summary: a synaptic vesicle. By contrast, P2Y receptors are activated by low concentrations of ATP (in the nM range... + wave propagation in astrocytes is another slow response mediated by P2Y receptor activation8,9 .Last... ACh-mediated transmission if P2X receptors are ... |
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Source: Lester, Henry - Division of Biology, California Institute of Technology |
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Collection: Biology and Medicine |
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| 35 | Muscarinic M3-receptors mediate cholinergic synergism of mitogenesis in | ||
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Summary: for the mitogenic contribution of muscarinic receptor stimulation. The p42/p44 mitogen activated protein kinase... -dependent mechanisms [16]. Moreover, the M3-receptor subtype activates protein kinase C (PKC), which may lead to p42/p... MAPK pathway induced by carbachol [18]. This ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 36 | Hetero-oligomerization between GABAA and GABAB Receptors Regulates GABAB Receptor Trafficking* | ||
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Summary: provided by Robert Lefkowitz (Duke University Medical Center). 1A-, 1B-, and 1D-adrenergic receptor... receptors in regulating each other's binding prop- erties (2325) and activity (24, 2629). In recent years... , 1st 3 lanes). Conversely, GST alone did not ... |
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Source: Teissére, Jeremy Alden - Biology Department, Muhlenberg College |
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Collection: Biology and Medicine |
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| 37 | Hetero-oligomerization between GABAA and GABAB Receptors Regulates GABAB Receptor Trafficking* | ||
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Summary: (Duke University Medical Center). 1A-, 1B-, and 1D-adrenergic receptor constructs were kindly provided... receptors in regulating each other's binding prop- erties (2325) and activity (24, 2629). In recent years... with an antibody against the 2 subunit (Fig. 5A, ... |
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Source: Hall, Randy A - Department of Pharmacology, Emory University |
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Collection: Biology and Medicine |
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| 38 | The serotonergic system The Serotonergic System | ||
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Summary: shown that 5-HT2A receptor increases cAMP in A1A1 adrenal cells by the intermediary action of calmodulin... animals were insensitive to the hyperlocomotor effects of the 5-HT1A/1B receptor agonist RU... ), Src kinase, and ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 39 | Research Article Northern Ring Conformation of Methanocarba-Adenosine | ||
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Summary: ** ** 0.5 nA 1 s B C D ATP 3 µM MRS 2312 3 µM MRS 2340 3 µM Fig. 3. Activity of methanocarba... for Activation of P2X Receptors Philip M. Dunn,1n Hak Sung Kim,2 Kenneth A. Jacobson,3 and Geoffrey Burnstock1 1... produces agonists with widely differing activities ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 40 | The structure of active opsin as a basis for identification of GPCR agonists by dynamic homology modelling and virtual screening assays | ||
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Summary: modelling and virtual screening assays Michael Schneider a,1 , Steffen Wolf a,b , Jürgen Schlitter a , Klaus... of opsin [15] and most recently structural models of active conformations of the b2-adrenergic receptor (B2... AR) [1618], the agonist-bound b1-adrenergic receptor [19] and a ... |
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Source: Gerwert, Klaus - Fakultät für Biologie, Ruhr-Universität Bochum |
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Collection: Biology and Medicine |
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| 41 | Serotonin is a biogenic amine that activates a large and heterogeneous family of receptors that are widely | ||
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Summary: Serotonin is a biogenic amine that activates a large and heterogeneous family of receptors... equivalent binding sites, although these may not all need to be occupied to efficiently activate the receptor... ). Furthermore, the role of 5-HT3 receptors in modulating ... |
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Source: Traynelis, Stephen F. - Department of Pharmacology, Emory University |
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Collection: Biology and Medicine |
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| 42 | 5-HT Receptors and the Neuromodulatory Control of | ||
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Summary: ................................................................................................ 9 3.2 5-HT1A/1B receptors facilitate the induction of long-term depression... the low expression of 5-HT2A/2C receptors in the dorsal horn (see Section 2.2.2). 3.2 ... |
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Source: Hochman, Shawn - Department of Physiology, Emory University |
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Collection: Biology and Medicine |
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| 43 | General discussion 1. Neurobiological consequences of chronic partial sleep deprivation | ||
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Summary: desensitization of the adenosine A1 receptor system, but did not result in a desensitized serotonin-1A signalling... to sleep. This forced activity control group did not show the desensitization in serotonin-1A receptor... of the muscarinic cholinergic receptors, ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 44 | Progress in Neurobiology 70 (2003) 387407 Kainate receptors and synaptic transmission | ||
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Summary: , GABAB, muscarinic or adenosine A1 receptor activation, suggesting that ATPA may act directly... M CGP55845) or adenosine A1 (0.1 M DPCPX) receptors. Similar results were obtained by Kamiya... - sure to the GABAB receptor ... |
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Source: Huettner, James E. - Department of Cell Biology and Physiology, Washington University in St. Louis |
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Collection: Biology and Medicine |
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| 45 | Olfactory receptor trafficking to the plasma membrane C. F. Bush and R. A. Hall* | ||
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Summary: activity of the receptors accompanied by persistent internalization. In accordance with this scenario... 12, 17-4, 3A1, 52E2, 51I2, 2AG1, 52B4, 4C15, mouse I7) with Hsc70t in HEK-293 cells significantly... , M. T. (2003) Activation of purinergic receptor subtypes ... |
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Source: Hall, Randy A - Department of Pharmacology, Emory University |
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Collection: Biology and Medicine |
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| 46 | REVIEW ARTICLE Chemokine receptors and other G protein-coupled receptors | ||
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Summary: D, Zhang L, et al. Heterologous expression of the adenosine A1 receptor in transgenic mouse retina... to understanding ligand binding, activation and function as co-receptors during viral entry. Keywords CCR5 and CXCR... , Hamm HE. Heterotrimeric G protein activation ... |
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Source: Palczewski, Krzysztof - Department of Pharmacology, Case Western Reserve University |
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Collection: Biology and Medicine |
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| 47 | Associate editor: A.L. Morrow Regulation of GABAA receptor trafficking, channel activity, | ||
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Summary: postsynaptically concentrated GABAA receptor subtypes identified to date, most commonly in association with the a1... -deficient mice (Gu¨n- ther et al., 1995). Clustering of a1 and a2 subunit-containing receptor subtypes is reduced... ;rescues clustering of ... |
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Source: Luscher, Bernhard - Department of Biology, Pennsylvania State University |
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Collection: Biology and Medicine |
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| 48 | Regulation of Neurotransmitter Release by Metabotropic Glutamate Receptors | ||
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Summary: demonstrated that the activation of mGlu receptors can modulate the activity of Ca2 or K channels, or interfere... activated by 3,5-dihydroxyphenyl- glycine (DHPG) or quisqualate. In contrast, the remain- ing receptors... potent at group I mGlu receptors, also has ... |
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Source: Alford, Simon - Department of Biological Sciences, University of Illinois at Chicago |
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Collection: Biology and Medicine |
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| 49 | AMPA receptor desensitization mutation results in severe developmental phenotypes and early | ||
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Summary: receptor subunits GluA1 and GluA2 was decreased, whereas NMDA receptor protein expression was increased... from the four re- ceptor subunits GluA1GluA4 (GluR14) (1). These recep- tors are activated... in the amount of ... |
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Source: Contractor, Anis - Department of Physiology, Northwestern University |
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Collection: Biology and Medicine |
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| 50 | Conclusions, Perspectives, | ||
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Summary: the motility, suggesting freezing as another factor in receptor activation. Further study also showed... of the receptor. The simulations have led to a new model regarding the activation of the receptor. Besides... , the simulations allowed discrimination between the states of the ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 51 | TRENDS in Pharmacological Sciences Vol.22 No.4 April 2001 http://tips.trends.com 0165-6147/01/$ see front matter 2001 Elsevier Science Ltd. All rights reserved. PII: S0165-6147(00)01643-6 | ||
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Summary: , four subtypes of adenosine (P1) receptors were cloned [A1 , A2A , A2B and A3 (Ref. a)]. P2X receptor... breakdown to adenosine, it acts as a prejunctional inhibitor of transmission via adenosine A1 receptors... Antagonists Transduction ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 52 | Bulletin of Mathematical Biology (2008) 70: 15251569 DOI 10.1007/s11538-008-9321-6 | ||
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Summary: directly interact with the receptors. To bring about tumbling, the receptors activate Che... the receptor methylation state which mediates adaptation by reducing the ability of the receptors to activate... to demethylate the receptors counter- ... |
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Source: Maini, Philip K. - Centre for Mathematical Biology & Mathematical Institute, University of Oxford |
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Collection: Mathematics ; Biology and Medicine |
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| 53 | International Union of Pharmacology LVIII: Update on the P2Y G Protein-Coupled Nucleotide Receptors | ||
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Summary: . . 286 3. Voltage-activated channels regulated by P2Y receptors... . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . . 287 4. Activation or inactivation of G protein-gated K channels by P2Y receptors... . . . . . . . . . . . . . . . . . . . . . . . . . . ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 54 | UCB Pharma research day--25 October 2007 `Glia-neuron interactions and purinergic receptors | ||
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Summary: . In the early 1990s, P1 and P2 receptors were cloned and characterised: four P1 receptor subtypes (A1, A2A, A2B... in dentate granule cells (CG). P2Y1R signalling in astrocytes activates presynaptic NMDA receptors via... by activating ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 55 | Although it has been known for more than half a century that extracellular purines, and specifically ATP, can affect | ||
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Summary: of the TGF response. Pharmacological blockade of the adenosine A1 receptor inhibits, and A1 recep- tor... of specific P2 receptor activation have been limited by the need to define different P2 receptors pharma... , ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 56 | Diinosine pentaphosphate: an antagonist which discriminates between recombinant P2X3 and P2X2/3 receptors and between two | ||
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Summary: pentaphosphate (Ip5I) is a very potent antagonist at recombinant P2X1 receptors (pA2, 8.2) and is quite active... the antagonist activity of Ip5I at the recombinant heteromeric P2X2/3 receptor. We have then compared... and P2X3 transcripts, the transient current due to activation of ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 57 | Purinergic receptors modulate MAP kinases and transcription factors that control microglial inflammatory gene expression | ||
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Summary: demonstrated that P2 purinergic receptor activation by ATP decreases cytokine, nitric oxide (NO), inducible... microglia with TNF-a and the P2X7 receptor agonist BzATP attenuates p38 MAPK activation, this is not true... concentrations of ATP that stimulate P2X7 receptor ... |
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Source: Kalil, Ronald E. - Neuroscience Training Program & W.M. Keck Laboratory for Biological Imaging, University of Wisconsin at Madison |
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Collection: Biology and Medicine |
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| 58 | Characterization of Interactions between Death Receptor 5 and its Ligand TRAIL | ||
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Summary: are indicated by colours. The DR5 N1 domain is shown in green. A1 domains are shown in orange/red/magenta and B2... preventing it from activating the death receptors. Two of the decoy receptors are membrane bound, namely... membrane proteins, with the exception of OPG. The ... |
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Source: Groningen, Rijksuniversiteit - Centre for Ecological and Evolutionary Studies, Department of Marine Benthic Ecology and Evolution, |
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Collection: Biology and Medicine ; Environmental Sciences and Ecology |
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| 59 | PERSPECTIVE Orphan nuclear receptors--new ligands | ||
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Summary: steroid receptors. Prominently inducible members of the rodent P450 3A gene family (CYP3A1, CYP3A2, CYP3A... - tochrome P-450 3A1 by dexamethasone and the antigluco- New orphan receptor ligands GENES & DEVELOPMENT 3153... to the known ... |
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Source: Blumberg, Bruce - Department of Developmental and Cell Biology, University of California, Irvine |
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Collection: Biology and Medicine |
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| 60 | Diabetes Metab . Author manuscript Cannabinoid receptors as novel therapeutic targets for the management of | ||
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Summary: experimental and clinical data indicate that peripheral activation of cannabinoid CB1 receptors promotes... in several countries for the management of chemotherapy-induced nausea and vomiting ( ) and rimonabant, a1... -Hyiaman D , Park O . Paracrine activation of hepatic CB1 ... |
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Source: Ecole Polytechnique, Centre de mathématiques |
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Collection: Mathematics |
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| 61 | Review article Eph receptorephrin bidirectional signals that target Ras and Rho proteins | ||
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Summary: factor, affects the activities of these proteins. Stimulation of EphA receptors by ephrin-A1 in T cells... and mediates RhoA activation in rat vascular smooth muscle cells stimulated with ephrin-A1 Fc [53... effects mediated by ... |
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Source: Chin-Sang, Ian - Department of Biology, Queen's University (Kingston) |
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Collection: Biology and Medicine |
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| 62 | Perspectives in Pharmacology P2 Purinergic Receptors: Modulation of Cell Function and | ||
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Summary: this response. AMP gives rise to adenosine, which acti- vates the various P1 receptors (A1, A2A, A2B, A3... ) that are rapidly activated and desensitized; group 2 includes P2X2, P2X4, P2X5, and P2X6 receptors that have lower... with the excitatory actions of ATP on nerve cells. Adenosine ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 63 | TheJournalofHistochemistry&Cytochemistry The Histochemical Society, Inc. 0022-1554/05/$3.30 1273 | ||
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Summary: ; Figures 1A, 1D, and 1F). Most P2X1, P2X3, P2X4, and P2X6 receptor staining was detected in small... to be activated by extracellular nucleotides. These receptors share be- tween 25% and 55% identity (at the amino... ) and modu- lation of the capsaicin receptor, TRPV1 ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 64 | JOURNAL OF VIROLOGY, 0022-538X/99/$04.00 0 | ||
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Summary: a Juxtamembrane Negative Charge for Activation of the Platelet-Derived Growth Factor Receptor and Transformation... ) receptor through transmembrane and juxtamembrane interactions, leading to sustained receptor activation... to transform C127 mouse fibroblasts and to bind to and induce ... |
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Source: DiMaio, Daniel - Departments of Genetics & Molecular Biophysics and Biochemistry, Yale University; Klein, Ophir - Departments of Orofacial Sciences & Pediatrics, University of California at San Francisco; Smith, Steven O.- Department of Biochemistry and Cell Biology, SUNY at Stony Brook |
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Collection: Biology and Medicine |
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| 65 | Pharmacological characterization of serotonin receptor subtypes modulating primary aerent input to deep dorsal horn neurons in | ||
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Summary: University, Atlanta, Georgia, GA 30322, U.S.A. 1 Spinal cord slices and whole-cell patch clamp recordings... . This action was probably mediated by 5-HT1A receptor activation, since it occurred in the presence of the 5-HT... , suggesting that there is sucient endogenous 5-HT to tonically ... |
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Source: Hochman, Shawn - Department of Physiology, Emory University |
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Collection: Biology and Medicine |
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| 66 | Progesterone, but Not Progesterone-Independent Activation of Progestin Receptors by a Mating | ||
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Summary: Progesterone, but Not Progesterone-Independent Activation of Progestin Receptors by a Mating... cervical stimulation (VCS) can influence sexual behavior by activating pro- gestin receptors in the absence... that progestin receptors are activated by VCS at this time. ... |
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Source: Blaustein, Jeffrey D. - Center for Neuroendocrine Studies, University of Massachusetts at Amherst |
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Collection: Biology and Medicine |
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| 67 | Cys-loop receptors: new twists and turns | ||
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Summary: been observed as a result of M2M3 linker region mutations in glycine receptors [4345], nicotinic a1... of naturally occurring pathological mutations in the M2M3 linker region of the glycine receptor a1 subunit [43... ,44] and the nicotinic ACh ... |
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Source: Lester, Henry - Division of Biology, California Institute of Technology |
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Collection: Biology and Medicine |
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| 68 | Functional Properties of Perigeniculate Inhibition of Dorsal Lateral Geniculate Nucleus Thalamocortical Neurons In Vitro | ||
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Summary: in micropipette) to lamina A1, the glutamate applications to the PGN are repeated and activate slow IPSPs... , with the strong activation of GABAB receptors requiring an intense, simultaneous discharge of a number of PGN... - tially through the activation of GABAA ... |
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Source: McCormick, David - Department of Neurobiology, Yale University |
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Collection: Biology and Medicine |
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| 69 | Function and structure in glycine receptors and some of their relatives | ||
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Summary: to nicotinic receptors, observations on glycine homomeric a1 receptors [29,30] cannot be fitted well... -channel methods is the glycine a1 receptor [29,30]. It seems likely that this homomeric pentamer would... mechanism of ... |
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Source: Colquhoun, David - Department of Pharmacology, University College London |
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Collection: Biology and Medicine |
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| 70 | Purinergic signalling: therapeutic potential* GEOFFREY BURNSTOCK | ||
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Summary: receptors were cloned, namely A1, A2A, A2B and A3 and in 1985, Burnstock and Kennedy proposed a basis... -prolonging role in heart failure; increased expression or activation of these ATP- stimulated receptor channels... suggested that resultant P2X7 receptor ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 71 | ORIGINAL ARTICLE Cells in Behaviourally Relevant Brain Regions Coexpress Nuclear Receptor | ||
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Summary: ). Steroid receptor coactivator-1 (SRC-1, also known as NCoA-1), was the first coactivator of steroid... into the active form (10). The activated receptors dimerise and preferentially bind to steroid response elements... -dependent transcriptional ... |
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Source: Tetel, Marc J. - Department of Biological Sciences, Wellesley College |
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Collection: Biology and Medicine |
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| 72 | Bruce N. Cronstein, MD You Are Not Arthur Conan Doyle | ||
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Summary: Data "Adenosine A1 receptor activation stimulates SREBP1 translocation... problem. Moreover, the demonstration that adenosine A1 receptors may play... by either an adenosine ... |
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Source: Wang, Da-Neng - Skirball Institute of Biomolecular Medicine & Department of Cell Biology, New York University |
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Collection: Biology and Medicine |
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| 73 | 2001 Wiley-Liss, Inc. DRUG DEVELOPMENT RESEARCH 52:110 (2001) | ||
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Summary: were cloned, namely, A1, A2A, A2B, and A3 [Ralevic and Burnstock, 1998]. P2X Receptor Family P2X... :246254. Vainio M, Törnquist K. 2000. The role of adenosine A1 receptors in the ATP-evoked Ca2+ response in rat... fibers are activated via P2X3 ... |
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|
Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 74 | Page 1 Biographical Sketch Format Page Principal Investigator/Program Director (Last, First, Middle): Ingraham, Holly A., Ph.D. | ||
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Summary: receptor mediated rapid signaling and nuclear actions in breast cancer cell models: role of mitogen-activated... receptors upregulate Wnt-1 to induce EGFR transactivation and c- Src dependent Sustained Activation of Erk1... , E.J. and C.A. Lange, Temporal Activation of Erk 1/2 MAPK by ... |
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|
Source: Ingraham, Holly - Department of Physiology, University of California at San Francisco |
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Collection: Biology and Medicine |
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| 75 | Research Signpost 37/661 (2), Fort P.O., Trivandrum-695 023, Kerala, India | ||
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Summary: by the selective A1 receptor antagonist 8- cyclopentyl-1,3-dipropylxanthine (DPCPX). The ecto-ATPase inhibitor (ARL... then activates P2X3 and/or P2X2/3 receptors on subepithelial sensory nerve plexuses to relay messages to the CNS... of the bladder and this activity ... |
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Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 76 | Neurons respond to a variety of attractive and repulsive guid-ance cues to navigate to their targets1. Genetic, biochemical and | ||
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Summary: midline crossing. When comm is absent, review Ligand binding FNIII EPH RECEPTORS EphA18, EphB16 VAB-1... Plexin-A14,B13,C1,D1 PLX-1,2 Plexin-A,B NEUROPILIN Neuropilin-1,2 Ligands Receptors Responses TSP... A receptors. Cell 99, ... |
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Source: Bargmann, Cori - Laboratory of Neural Circuits and Behavior, Rockefeller University |
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Collection: Biology and Medicine |
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| 77 | PC PE PS PI SPM GangChol | ||
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Summary: of the EGF receptor is increased. #12;Cholesterol depletion also leads to the activation of MAP kinase... suppresses the activity of this receptor and is probably important in maintaining the EGF receptor... signaling, including the EGF receptor, has led to the ... |
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Source: Pike, Linda J. - Department of Biochemistry and Molecular Biophysics, Washington University in St. Louis |
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Collection: Biology and Medicine |
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| 78 | Mode of receptor binding and activation by plasminogen-related growth factors | ||
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Summary: Hypothesis Mode of receptor binding and activation by plasminogen-related growth factors Maria... domain enzymatic activity and became ligands for cell surface tyrosine kinase receptors... , low affinity for HGF), monomeric ligand induces receptor dimerization and ... |
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|
Source: Wlodawer, Alexander - Macromolecular Crystallography Laboratory, National Cancer Institute |
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Collection: Chemistry ; Biology and Medicine |
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| 79 | FAST KINETIC MODELS FOR SIMULATING AMPA, NMDA, | ||
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Summary: underlyingsynaptic transmission. Particular receptor types have been identi ed and their activation kinetics... the kinetics of activation of these receptors. It was shown that introducing simplifying assumptions leads... and neuromodulation. Synaptic receptors ... |
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|
Source: Boahen, Kwabena - Department of Bioengineering, Stanford University; Destexhe, Alain - Unité de Neurosciences Intégratives et Computationnelles, CNRS |
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Collection: Biology and Medicine ; Computer Technologies and Information Sciences |
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| 80 | The International Journal of Biochemistry & Cell Biology 35 (2003) 130134 Molecules in focus | ||
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Summary: collectively termed ephrins were subsequently identified that could bind Eph family receptors and activate... A RTKs (EphA1A8) promiscuously interact with five A-ephrins (ephrinA1A5), that are attached to the cell... signaling is unique in that both the ligand and ... |
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|
Source: Chin-Sang, Ian - Department of Biology, Queen's University (Kingston) |
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Collection: Biology and Medicine |
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| 81 | Activation and block of recombinant GABAA receptors by pentobarbitone: a single-channel study | ||
|
Summary: that recombinant a1b2g2L GABA receptors transiently expressed in HEK cells can be activated by PB. High... -channel conductance of the a1b2g2 GABA receptor is similar when the receptors are activated by ... |
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|
Source: Steinbach, Joe Henry - Washington University Pain Center & Department of Anesthesiology, Washington University in St. Louis |
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Collection: Biology and Medicine |
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| 82 | This article appeared in a journal published by Elsevier. The attached copy is furnished to the author for internal non-commercial research | ||
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Summary: activators. A variety of studies in cell lines reveal that nuclear receptor coregulators are critical... receptors, which are members of the steroid/nuclear receptor superfamily of transcriptional activators [111... receptor coregulators enhance (coactivators) or ... |
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|
Source: Tetel, Marc J. - Department of Biological Sciences, Wellesley College |
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Collection: Biology and Medicine |
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| 83 | EDITED B'r' Bertha K. Madras Harvard Medical School | ||
|
Summary: , and serotonin (5-HT3) receptors. Currently, 12 neu- ronal nAChR subunits have been identified (a2--a1 0 and 132... effects by binding to and activating neuronal nicotinic acetylcholine receptors (nAChRs) in the brain... . Nicotinic receptors are pentameric ... |
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|
Source: Lester, Henry - Division of Biology, California Institute of Technology |
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Collection: Biology and Medicine |
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| 84 | An aplysia dopamine1-like receptor: molecular and functional characterization | ||
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Summary: , central nervous system, constitutive activity, dopamine, G-protein- coupled receptor. J. Neurochem. (2006... activity. Based on their sequence similarity and pharmacological profile, the DA receptors in vertebrate... D2-like receptors inhibit adenylyl cyclase and ... |
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|
Source: Byrne, John H. - Department of Neurobiology and Anatomy, University of Texas Medical School at Houston |
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Collection: Biology and Medicine |
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| 85 | Distinct Structural Changes in the GABAA Receptor Elicited by Pentobarbital and GABA | ||
|
Summary: complicates the interpretation, the results in a1b2K274Cg2 receptors offer an example where GABA activation... receptors. a1b2g2N135C expressed well; when labeled with TMRM, however, this receptor showed no changes... showed ... |
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|
Source: Kalil, Ronald E. - Neuroscience Training Program & W.M. Keck Laboratory for Biological Imaging, University of Wisconsin at Madison |
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Collection: Biology and Medicine |
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| 86 | REVIEW ARTICLE Nuclear Receptor Coactivators: Essential Players for Steroid Hormone | ||
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Summary: of the steroid / nuclear receptor superfamily of transcriptional activators (1, 2). Receptors for oestrogens (ER... for modulating the transcriptional activity of ER and PR, as well as other nuclear receptors. Although ER and PR... -terminal ligand binding domain (1, 2). In general, ... |
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|
Source: Tetel, Marc J. - Department of Biological Sciences, Wellesley College |
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Collection: Biology and Medicine |
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| 87 | SYNERGISTIC SEDATIVE EFFECTS OF NORADRENERGIC a1-AND b-RECEPTOR BLOCKADE ON FOREBRAIN ELECTROENCEPHALOGRAPHIC AND | ||
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Summary: that was associated with decreased behavioral activity; (iii) combined a1- and b-receptor blockade elicits... and/or behavioral indices of arousal/waking.9,29 a1-Receptors also exert an activational influence... on beha- ... |
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|
Source: Kalil, Ronald E. - Neuroscience Training Program & W.M. Keck Laboratory for Biological Imaging, University of Wisconsin at Madison |
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Collection: Biology and Medicine |
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| 88 | Introduction In 1987, a receptor was identified in a search for tyrosine | ||
|
Summary: carcinoma cell line from which its cDNA was isolated. Today, 16 receptors (EphA1-10 and EphB1-6) and 9... system and constitutively binds the kinase domain of EphA receptors. Interestingly, ephrin-A1 treatment... factor Tcf-4, which is activated ... |
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|
Source: Chin-Sang, Ian - Department of Biology, Queen's University (Kingston) |
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Collection: Biology and Medicine |
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| 89 | Z .European Journal of Pharmacology 405 2000 7388 www.elsevier.nlrlocaterejphar | ||
|
Summary: receptor within a1 circumscribed time window yielded greater potentiation than simultaneous exposure... of potentiation.1 Pre-exposure of vasopressin V receptor agonist for 60 s resulted in a1 75% potentiation... constraints of vasopressin-induced potentiation ... |
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|
Source: Brinton, Roberta Diaz - Laboratory for Neuroscience Research & School of Pharmacy, University of Southern California |
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Collection: Biology and Medicine |
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| 90 | Current Topics in Medicinal Chemistry 2004, 4, 793-803 793 1568-0266/04 $45.00+.00 2004 Bentham Science Publishers Ltd. | ||
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Summary: receptor family. The kinetics of activation, inactivation and deactivation also vary considerably amongst P... and operational profiles. In response to nucleotide activation, recombinant P2Y receptors either activate... are activated by all triphosphate nucleotides. ... |
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|
Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 91 | Central Projections of Auditory Receptor Neurons of Crickets | ||
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Summary: * Department of Biology, McGill University, Montreal, Quebec H3A1B1, Canada ABSTRACT We describe the central... . Pollack, Dept. of Biology, McGill Univer- sity, 1205 Avenue Docteur Penfield, Montreal, QC H3A1B1, Canada... Central Projections of Auditory Receptor Neurons of Crickets KAZUO ... |
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|
Source: Pollack, Gerald - Department of Biology, McGill University |
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Collection: Environmental Sciences and Ecology |
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| 92 | *National Institute of Child Health and Human | ||
|
Summary: concentra- tions of adenosine activate the A1 receptor expressed on neutrophils, whereas high concentrations... - quently co-expressed in single hippocampal pyramidal neurons97 . A1 receptor activation can inhibit... released ... |
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|
Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 93 | The EMBO Journal vol.10 no.4 pp.845-855, 1991 Activation of the platelet-derived growth factor receptor | ||
|
Summary: , a metabolic precursor as well as the mature form of the receptor is activated by E5 transformation. Activation... stimulation in this system. Moreover, activation of the receptor by addition of PDGF or the v-sis gene... that the PDGF receptor is an important ... |
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|
Source: DiMaio, Daniel - Departments of Genetics & Molecular Biophysics and Biochemistry, Yale University |
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Collection: Biology and Medicine |
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| 94 | Special issue: Allosterism and Collateral Efficacy Conformational complexity of | ||
|
Summary: Scheer, A. et al. (1997) The activation process of the a1B-adrenergic receptor: potential role... histamine receptor [20], the a1b adrenoceptor [21,22] and the angiotensin (AT1) receptor [23]. My co... . Pharmacol. 57, ... |
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|
Source: Kobilka, Brian - Department of Molecular and Cellular Physiology, Stanford University |
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Collection: Biology and Medicine |
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| 95 | Orphan nuclear receptors adopted by crystallography Holly A Ingraham1 | ||
|
Summary: protein fold that consists of an a-helical bundle (a1a12) with a small number of b-strands (Figure 1b... binds and result in co-activator recruit- ment through a nuclear receptor interaction box (NR box... this model applies to all nuclear receptors including those that exhibit ... |
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|
Source: Ingraham, Holly - Department of Physiology, University of California at San Francisco |
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|
Collection: Biology and Medicine |
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| 96 | Role of delivery and trafficking of d-opioid peptide receptors in opioid | ||
|
Summary: activate MOP receptors and produce potent spinal analgesia. Among the agents used in pain treatment, opioid... receptors are internalized and processed in the degradation pathway after being activated in this way [14... attenuation of signaling. In general terms, it is accepted that ... |
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|
Source: Tian, Weidong - Institute of Biochemistry and Cell Biology, Shanghai Institute of Biological Sciences |
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Collection: Biology and Medicine |
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| 97 | Bovine Papillomavirus E5 Protein Induces the Formation of Signal Transduction Complexes Containing Dimeric Activated | ||
|
Summary: Dimeric Activated Platelet-derived Growth Factor Receptor and Associated Signaling Proteins* (Received... (PDGF) recep- tor, resulting in constitutive activation of the receptor and cell growth transformation... , activated PDGF receptor complexes were separated from ... |
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|
Source: DiMaio, Daniel - Departments of Genetics & Molecular Biophysics and Biochemistry, Yale University |
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Collection: Biology and Medicine |
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| 98 | Mapping convulsants' binding to the GABA-A receptor chloride ionophore: A proposed model for channel binding sites | ||
|
Summary: to eight families: a16, b13, g13, d, e, p, u and r13) around the ionophore (Baumann et al., 2001, 2002... ) modulating the receptor activity. Binding of GABA opens up a ClÀ channel, leading to neuronal inhibition... of the ability to inhibit different ionotropic receptors by ... |
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|
Source: Kalueff, Allan V. - Department of Pharmacology, Tulane University |
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Collection: Biology and Medicine |
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| 99 | The FASEB Journal express article 10.1096/fj.03-1175fje. Published online July 1, 2004. Purinoceptor expression in regenerating skeletal muscle in | ||
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Summary: is an important extracellular signaling molecule mediating its effects by activation of P2X and P2Y receptors. P2... regeneration. The P2X5 and P2Y1 receptors were expressed first on activated satellite cells, and the P2Y1... receptors (5). P2Y receptors are G ... |
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|
Source: Burnstock, Geoffrey - Autonomic Neuroscience Centre, University College London |
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Collection: Biology and Medicine |
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| 100 | Behaioural Pharmacology 2001; 00:1 10 REVIEW Serotonin receptors in mood disorders: a combined1A | ||
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Summary: , a1A temporal modulation of the transcriptional activity of the 5-HT1A receptor is achieved... transcriptional activation at both pre-1A 1A and postsynaptic sites; tTA Rescue: CamKII tTA rescues receptor... lines of evidence ... |
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|
Source: Sibille, Etienne - Center for the Neural Basis of Cognition & Department of Psychiatry, University of Pittsburgh |
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Collection: Biology and Medicine |
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